HYPOTHALAMIC, PITUITARY AND UTERINE CYTOPLASMIC AND NUCLEAR ESTROGEN-RECEPTORS AND THEIR RELATIONSHIP TO THE SERUM CONCENTRATION OF TAMOXIFEN AND ITS METABOLITE, 4-HYDROXYTAMOXIFEN, IN THE OVARIECTOMIZED RAT

被引:26
作者
BOWMAN, SP [1 ]
LEAKE, A [1 ]
MORRIS, ID [1 ]
机构
[1] UNIV MANCHESTER, DEPT PHARMACOL MAT MED & THERAPEUT, MANCHESTER M13 9PT, LANCS, ENGLAND
关键词
D O I
10.1677/joe.0.0940167
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:167 / 175
页数:9
相关论文
共 26 条
[1]   MEASUREMENT OF TAMOXIFEN IN SERUM BY THIN-LAYER DENSITOMETRY [J].
ADAM, HK ;
GAY, MA ;
MOORE, RH .
JOURNAL OF ENDOCRINOLOGY, 1980, 84 (01) :35-42
[2]  
ADAM HK, 1979, BIOCHEM PHARMACOL, V27, P144
[3]  
BORGNA JL, 1981, J BIOL CHEM, V256, P859
[4]   HIGH-AFFINITY BINDING TO THE ESTROGEN-RECEPTOR OF [4-HYDROXYTAMOXIFEN-H-3, AN ACTIVE ANTI-ESTROGEN METABOLITE [J].
BORGNA, JL ;
ROCHEFORT, H .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1980, 20 (01) :71-85
[5]   TIME-RELATED EFFECTS OF EN-CLOMIPHENE UPON CENTRAL AND PERIPHERAL ESTROGEN TARGET TISSUES AND CYTOPLASMIC-RECEPTORS [J].
BOWMAN, SP ;
LEAKE, A ;
MORRIS, ID .
JOURNAL OF ENDOCRINOLOGY, 1981, 89 (01) :117-128
[6]   INVIVO EFFECT OF ANTI-ESTROGENS ON LOCALIZATION AND REPLENISHMENT OF ESTROGEN-RECEPTOR [J].
CAPONY, F ;
ROCHEFORT, H .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1975, 3 (03) :233-251
[7]  
CLARK JH, 1979, MONOGRAPHS ENDOCRINO, V14
[8]   EFFECTS OF ESTRADIOL AND THE ANTI-ESTROGEN TAMOXIFEN ON STEROID-HORMONE RECEPTOR CONCENTRATION AND NUCLEAR RIBONUCLEIC-ACID POLYMERASE ACTIVITIES IN RAT UTERI [J].
DAVIES, P ;
SYNE, JS ;
NICHOLSON, RI .
ENDOCRINOLOGY, 1979, 105 (06) :1336-1342
[9]   MODULATION OF RAT UTERINE STEROID-HORMONE RECEPTORS BY ESTROGEN AND ANTI-ESTROGEN [J].
DIX, CJ ;
JORDAN, VC .
ENDOCRINOLOGY, 1980, 107 (06) :2011-2020
[10]  
EDSALL JT, 1958, BIOPHYSICAL CHEM, V2