Thiazolo[4,3-c][1,4]benzodiazepines .1. Synthesis of amidine derivatives

被引：8

作者：

Gillard, AC

Rault, S

Boulouard, M

Robba, M

机构：

[1] Centre d'Etudes et de Recherche sur le Médicament de Normandie, U. F. R. des Sciences Pharmaceutiques, Caen, 14032

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1995年 / 32卷 / 06期

关键词：

D O I：

10.1002/jhet.5570320613

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Reactivity of 1,2,3,10,11,11a-hexahydro-5H-thiazolo[4,3-c][1,4]benzodiazepin-5-one-11-thione, and 1,2,3,10,11,11a-hexahydro-5H-thiazolo[4,3-c][1,4]benzodiazepine-5,11-dithione was evaluated against various amines. The synthetic pathways involved in these reactions which led to new thiazolo[4,3-c][1,4]benzodiazepine amidines are described.

引用

页码：1741 / 1745

页数：5

共 6 条

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