BIOCHEMICAL AND ENDOCRINE PROPERTIES OF A MECHANISM-BASED INHIBITOR OF AROMATASE

[1] THE STATUS OF OXYGEN-ATOMS IN THE REMOVAL OF C-19 IN ESTROGEN BIOSYNTHESIS [J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1981, (03) : 129 - 130

[2] INHIBITION OF TESTOSTERONE 5-ALPHA-REDUCTASE BY A PROPOSED ENZYME-ACTIVATED, ACTIVE SITE-DIRECTED INHIBITOR [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 95 (01) : 273 - 280

[3] INACTIVATION OF AROMATASE INVITRO BY 4-HYDROXY-4-ANDROSTENE-3, 17-DIONE AND 4-ACETOXY-4-ANDROSTENE-3, 17-DIONE AND SUSTAINED EFFECTS INVIVO [J]. STEROIDS, 1981, 38 (06) : 693 - 702

[4] AROMATASE INHIBITORS .4. REGRESSION OF HORMONE-DEPENDENT, MAMMARY-TUMORS IN THE RAT WITH 4-ACETOXY-4-ANDROSTENE-3,17-DIONE [J]. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1979, 10 (04) : 423 - 429

[5] BRODIE AMH, 1979, ENDOCRINOLOGY, V104, P118, DOI 10.1210/endo-104-1-118

[6] KINETIC PARAMETERS OF DRUG-METABOLIZING ENZYMES IN CA2+ - SEDIMENTED MICROSOMES FROM RAT-LIVER [J]. BIOCHEMICAL PHARMACOLOGY, 1972, 21 (24) : 3249 - +

[7] COVEY DF, 1981, J BIOL CHEM, V256, P1076

[8] ENZYME-GENERATED INTERMEDIATES DERIVED FROM 4-ANDROSTENE-3,6,17-TRIONE AND 1,4,6-ANDROSTATRIENE-3,17-DIONE CAUSE A TIME-DEPENDENT DECREASE IN HUMAN PLACENTAL AROMATASE-ACTIVITY [J]. ENDOCRINOLOGY, 1981, 108 (04) : 1597 - 1599

[9] FISHMAN J, 1981, J BIOL CHEM, V256, P4466

[10] PURIFICATION AND CHARACTERIZATION OF ADRENODOXIN REDUCTASE FROM BOVINE ADRENAL-CORTEX [J]. BIOCHEMISTRY, 1975, 14 (07) : 1477 - 1484

[1] THE STATUS OF OXYGEN-ATOMS IN THE REMOVAL OF C-19 IN ESTROGEN BIOSYNTHESIS [J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1981, (03) : 129 - 130

[2] INHIBITION OF TESTOSTERONE 5-ALPHA-REDUCTASE BY A PROPOSED ENZYME-ACTIVATED, ACTIVE SITE-DIRECTED INHIBITOR [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 95 (01) : 273 - 280

[3] INACTIVATION OF AROMATASE INVITRO BY 4-HYDROXY-4-ANDROSTENE-3, 17-DIONE AND 4-ACETOXY-4-ANDROSTENE-3, 17-DIONE AND SUSTAINED EFFECTS INVIVO [J]. STEROIDS, 1981, 38 (06) : 693 - 702

[4] AROMATASE INHIBITORS .4. REGRESSION OF HORMONE-DEPENDENT, MAMMARY-TUMORS IN THE RAT WITH 4-ACETOXY-4-ANDROSTENE-3,17-DIONE [J]. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1979, 10 (04) : 423 - 429

[5] BRODIE AMH, 1979, ENDOCRINOLOGY, V104, P118, DOI 10.1210/endo-104-1-118

[6] KINETIC PARAMETERS OF DRUG-METABOLIZING ENZYMES IN CA2+ - SEDIMENTED MICROSOMES FROM RAT-LIVER [J]. BIOCHEMICAL PHARMACOLOGY, 1972, 21 (24) : 3249 - +

[7] COVEY DF, 1981, J BIOL CHEM, V256, P1076

[8] ENZYME-GENERATED INTERMEDIATES DERIVED FROM 4-ANDROSTENE-3,6,17-TRIONE AND 1,4,6-ANDROSTATRIENE-3,17-DIONE CAUSE A TIME-DEPENDENT DECREASE IN HUMAN PLACENTAL AROMATASE-ACTIVITY [J]. ENDOCRINOLOGY, 1981, 108 (04) : 1597 - 1599

[9] FISHMAN J, 1981, J BIOL CHEM, V256, P4466

[10] PURIFICATION AND CHARACTERIZATION OF ADRENODOXIN REDUCTASE FROM BOVINE ADRENAL-CORTEX [J]. BIOCHEMISTRY, 1975, 14 (07) : 1477 - 1484