4,5,6,7-TETRAHYDROISOTHIAZOLO[5,4-C]PYRIDIN-3-OL AND RELATED ANALOGS OF THIP - SYNTHESIS AND BIOLOGICAL-ACTIVITY

被引：39

作者：

KROGSGAARDLARSEN, P ^{[1
]}

MIKKELSEN, H ^{[1
]}

JACOBSEN, P ^{[1
]}

FALCH, E ^{[1
]}

CURTIS, DR ^{[1
]}

PEET, MJ ^{[1
]}

LEAH, JD ^{[1
]}

机构：

[1] AUSTRALIAN NATL UNIV,DEPT PHARMACOL,CANBERRA,ACT 2601,AUSTRALIA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1983年 / 26卷 / 06期

关键词：

D O I：

10.1021/jm00360a020

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：895 / 900

页数：6

共 32 条

[21] GABA AGONISTS - DEVELOPMENT AND INTERACTIONS WITH THE GABA RECEPTOR COMPLEX [J].

KROGSGAARDLARSEN, P ;

FALCH, E .

MOLECULAR AND CELLULAR BIOCHEMISTRY, 1981, 38 (AUG) :129-146

[22] GAMMA-AMINOBUTYRIC ACID AGONISTS, ANTAGONISTS, AND UPTAKE INHIBITORS - DESIGN AND THERAPEUTIC ASPECTS [J].

KROGSGAARDLARSEN, P .

JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (12) :1377-1383

[23] STRUCTURE-ACTIVITY STUDIES ON INHIBITION OF GABA BINDING TO RAT-BRAIN MEMBRANES BY MUSCIMOL AND RELATED COMPOUNDS [J].

KROGSGAARDLARSEN, P ;

JOHNSTON, GAR .

JOURNAL OF NEUROCHEMISTRY, 1978, 30 (06) :1377-1382

[24]

KROGSGAARDLARSEN P, 1979, EUR J MED CHEM, V14, P157

[25] MUSCIMOL ANALOGS .2. SYNTHESIS OF SOME BICYCLIC 3-ISOXAZOLOL ZWITTERIONS [J].

KROGSGAARDLARSEN, P .

ACTA CHEMICA SCANDINAVICA SERIES B-ORGANIC CHEMISTRY AND BIOCHEMISTRY, 1977, 31 (07) :584-588

[26] NEW CLASS OF GABA AGONIST [J].

KROGSGAARDLARSEN, P ;

JOHNSTON, GAR ;

LODGE, D ;

CURTIS, DR .

NATURE, 1977, 268 (5615) :53-55

[27] DIHYDROMUSCIMOL, THIOMUSCIMOL AND RELATED HETEROCYCLIC-COMPOUNDS AS GABA ANALOGS [J].

KROGSGAARDLARSEN, P ;

HJEDS, H ;

CURTIS, DR ;

LODGE, D ;

JOHNSTON, GAR .

JOURNAL OF NEUROCHEMISTRY, 1979, 32 (06) :1717-1724

[28] STRUCTURE AND BIOLOGICAL-ACTIVITY OF A SERIES OF CONFORMATIONALLY RESTRICTED ANALOGUES OF GABA [J].

KROGSGAARDLARSEN, P ;

JOHNSTON, GAR ;

CURTIS, DR ;

GAME, CJA ;

MCCULLOCH, RM .

JOURNAL OF NEUROCHEMISTRY, 1975, 25 (06) :803-809

[29] DEUTERIUM LABELING OF THE GABA AGONISTS THIP, PIPERIDINE-4-SULFONIC ACID AND THE GABA UPTAKE INHIBITOR THPO [J].

KROGSGAARDLARSEN, P ;

JOHANSEN, JS ;

FALCH, E .

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1982, 19 (05) :689-702

[30]

MORSELLI PL, 1981, NEUROTRANSMITTERS SE

← 1 2 3 4 →