STRUCTURAL FACTORS OF IMPORTANCE FOR 5-HYDROXYTRYPTAMINERGIC ACTIVITY - CONFORMATIONAL PREFERENCES AND ELECTROSTATIC POTENTIALS OF 8-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN (8-OH-DPAT) AND SOME RELATED AGENTS

被引：29

作者：

ARVIDSSON, LE

KARLEN, A

NORINDER, U

KENNE, L

SUNDELL, S

HACKSELL, U

机构：

[1] ASTR ALAB AB,RES & DEV LABS,COMP GRAPH UNIT,S-15185 SODERTALJE,SWEDEN

[2] UNIV STOCKHOLM,ARRHENIUS LAB,DEPT ORGAN CHEM,S-10691 STOCKHOLM,SWEDEN

[3] GOTHENBURG UNIV,DEPT STRUCT CHEM,S-40033 GOTHENBURG,SWEDEN

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1988年 / 31卷 / 01期

关键词：

D O I：

10.1021/jm00396a034

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：212 / 221

页数：10

共 62 条

[1]

Allinger N. L., 1980, QCPE, P395

[2] CONFORMATIONAL-ANALYSIS .130. MM2 - HYDROCARBON FORCE-FIELD UTILIZING V1 AND V2 TORSIONAL TERMS [J].

ALLINGER, NL .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1977, 99 (25) :8127-8134

[3]

Arvidsson L E, 1986, Prog Drug Res, V30, P365

[4] 8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)TETRALIN, A NEW CENTRALLY ACTING 5-HYDROXYTRYPTAMINE RECEPTOR AGONIST [J].

ARVIDSSON, LE ;

HACKSELL, U ;

NILSSON, JLG ;

HJORTH, S ;

CARLSSON, A ;

LINDBERG, P ;

SANCHEZ, D ;

WIKSTROM, H .

JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (08) :921-923

[5] 8-HYDROXY-2-(ALKYLAMINO)TETRALINS AND RELATED-COMPOUNDS AS CENTRAL 5-HYDROXYTRYPTAMINE RECEPTOR AGONISTS [J].

ARVIDSSON, LE ;

HACKSELL, U ;

JOHANSSON, AM ;

NILSSON, JLG ;

LINDBERG, P ;

SANCHEZ, D ;

WIKSTROM, H ;

SVENSSON, K ;

HJORTH, S ;

CARLSSON, A .

JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (01) :45-51

[6]

ARVIDSSON LE, IN PRESS J MED CHEM

[7] BICYCLIC AND TRICYCLIC ERGOLINE PARTIAL STRUCTURES - RIGID 3-(2-AMINOETHYL)PYRROLES AND 3-(2-AMINOETHYL)PYRAZOLE AND 4-(2-AMINOETHYL)PYRAZOLE AS DOPAMINE AGONISTS [J].

BACH, NJ ;

KORNFELD, EC ;

JONES, ND ;

CHANEY, MO ;

DORMAN, DE ;

PASCHAL, JW ;

CLEMENS, JA ;

SMALSTIG, EB .

JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (05) :481-491

[8] CONFORMATIONAL STUDY OF LYSERGIC-ACID AND ISO-LYSERGIC ACID DIALKYLAMIDES BY PROTON MAGNETIC-RESONANCE SPECTROSCOPY [J].

BAILEY, K ;

GREY, AA .

CANADIAN JOURNAL OF CHEMISTRY-REVUE CANADIENNE DE CHIMIE, 1972, 50 (23) :3876-3885

[9] MOLECULAR STRUCTURE OF LSD [J].

BAKER, RW ;

WEBER, HP ;

CHOTHIA, C ;

PAULING, P .

SCIENCE, 1972, 178 (4061) :614-&

[10]

BAKER RW, 1973, MOL PHARMACOL, V9, P23

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