STRUCTURAL FACTORS OF IMPORTANCE FOR 5-HYDROXYTRYPTAMINERGIC ACTIVITY - CONFORMATIONAL PREFERENCES AND ELECTROSTATIC POTENTIALS OF 8-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN (8-OH-DPAT) AND SOME RELATED AGENTS

被引：29

作者：

ARVIDSSON, LE

KARLEN, A

NORINDER, U

KENNE, L

SUNDELL, S

HACKSELL, U

机构：

[1] ASTR ALAB AB,RES & DEV LABS,COMP GRAPH UNIT,S-15185 SODERTALJE,SWEDEN

[2] UNIV STOCKHOLM,ARRHENIUS LAB,DEPT ORGAN CHEM,S-10691 STOCKHOLM,SWEDEN

[3] GOTHENBURG UNIV,DEPT STRUCT CHEM,S-40033 GOTHENBURG,SWEDEN

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1988年 / 31卷 / 01期

关键词：

D O I：

10.1021/jm00396a034

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：212 / 221

页数：10

共 62 条

[31]

JACKMAN LM, 1969, APPLICATIONS NMR SPE

[32]

JOHANSSON AM, 1986, MOL PHARMACOL, V30, P258

[33] C3-METHYLATED 5-HYDROXY-2-(DIPROPYLAMINO)TETRALINS - CONFORMATIONAL AND STERIC PARAMETERS OF IMPORTANCE FOR CENTRAL DOPAMINE RECEPTOR ACTIVATION [J].

JOHANSSON, AM ;

NILSSON, JLG ;

KARLEN, A ;

HACKSELL, U ;

SVENSSON, K ;

CARLSSON, A ;

KENNE, L ;

SUNDELL, S .

JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (07) :1135-1144

[34]

JOHANSSON AM, IN PRESS J MED CHEM

[35] CORRELATION BETWEEN ACTIVITY AND ELECTRONIC STATE OF HALLUCINOGENIC AMPHETAMINES [J].

KANG, S ;

GREEN, JP .

NATURE, 1970, 226 (5246) :645-&

[36] CONFORMATIONAL-ANALYSIS OF THE DOPAMINE-RECEPTOR AGONIST "5-HYDROXY-2-(DIPROPYLAMINO)TETRALIN AND ITS C(2)-METHYL-SUBSTITUTED DERIVATIVE [J].

KARLEN, A ;

JOHANSSON, AM ;

KENNE, L ;

ARVIDSSON, LE ;

HACKSELL, U .

JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (06) :917-924

[37] MECHANISM OF ACTION OF CHLORPROMAZINE [J].

KARREMAN, G ;

ISENBERG, I ;

SZENTGYORGYI, A .

SCIENCE, 1959, 130 (3383) :1191-1192

[38]

KIDRIC J, 1983, PERIOD BIOL, V85, P127

[39] DESCRIPTION OF STERIC RELATIONSHIPS ACROSS SINGLE BONDS [J].

KLYNE, W ;

PRELOG, V .

EXPERIENTIA, 1960, 16 (12) :521-523

[40] CONFORMATIONALLY RESTRICTED DOPAMINE CONGENERS - A MOLECULAR MECHANICS-BASED STUDY [J].

KOCJAN, D ;

HADZI, D .

JOURNAL OF PHARMACY AND PHARMACOLOGY, 1983, 35 (12) :780-785

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