MURAMYL PEPTIDE ANALOGS - SYNTHESIS OF A DEPSIPEPTIDE USING ORTHOGONAL SPPS

被引：4

作者：

CUNNINGHAM, BR

HANNAH, J

JONES, AB

机构：

[1] Department of Synthetic Chemical Research Merck Research Laboratories, Rahway, NJ 07065, R50G-146

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 51期

关键词：

D O I：

10.1016/0040-4039(94)88500-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A depsipeptide mimic of the cram-positive muramyl peptide was synthesized on resin using both Boc and Fmoc protection strategies. The depsipeptide unit is chemically and stereochemically compatible with both Boc and Fmoc chemistries and with HF cleavage conditions.

引用

页码：9517 / 9520

页数：4

共 9 条

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