RELATIVE AFFINITIES OF THE QUATERNARY NARCOTIC-ANTAGONIST, N-METHYL LEVALLORPHAN (SR-58002), FOR DIFFERENT TYPES OF OPIOID RECEPTORS

被引：7

作者：

BIANCHETTI, A

DRAGONETTI, M

GIUDICE, A

TARANTINO, A

FERRARESE, N

MANARA, L

APPELMANS, N

SIMON, EJ

机构：

[1] NYU,SCH MED,DEPT PSYCHIAT,NEW YORK,NY 10003

[2] NYU,SCH MED,DEPT PHARMACOL,NEW YORK,NY 10003

来源：

NEUROPEPTIDES | 1985年 / 5卷 / 4-6期

关键词：

D O I：

10.1016/0143-4179(85)90033-2

中图分类号：

R5 [内科学];

学科分类号：

1002 ; 100201 ;

摘要：

引用

页码：379 / 382

页数：4

共 11 条

[1] PHARMACOLOGICAL ACTIONS OF LEVALLORPHAN ALLYL BROMIDE (CM-32191), A NEW PERIPHERAL NARCOTIC-ANTAGONIST [J].

BIANCHETTI, A ;

GIUDICE, A ;

PICERNO, N ;

CARMINATI, P .

LIFE SCIENCES, 1982, 31 (20-2) :2261-2264

[2] QUATERNARY DERIVATIVES OF NARCOTIC-ANTAGONISTS - STEREOCHEMICAL REQUIREMENTS AT THE CHIRAL NITROGEN FOR INVITRO AND INVIVO ACTIVITY [J].

BIANCHETTI, A ;

NISATO, D ;

SACILOTTO, R ;

DRAGONETTI, M ;

PICERNO, N ;

TARANTINO, A ;

MANARA, L ;

ANGEL, LM ;

SIMON, EJ .

LIFE SCIENCES, 1983, 33 :415-418

[3] LEVALLORPHAN METHYL-IODIDE (SR-58002), A POTENT NARCOTIC-ANTAGONIST WITH PERIPHERAL SELECTIVITY SUPERIOR TO THAT OF OTHER QUATERNARY COMPOUNDS [J].

DRAGONETTI, M ;

BIANCHETTI, A ;

SACILOTTO, R ;

GIUDICE, A ;

FERRARESE, N ;

CATTANEO, C ;

MANARA, L .

LIFE SCIENCES, 1983, 33 :477-480

[4] KINETIC PARAMETERS OF NARCOTIC AGONISTS AND ANTAGONISTS WITH PARTICULAR REFERENCE TO N-ALLYLNOROXYMORPHONE (NALOXONE) [J].

KOSTERLITZ, HW ;

WATT, AJ .

BRITISH JOURNAL OF PHARMACOLOGY, 1968, 33 (02) :266-+

[5] THE BINDING SPECTRUM OF NARCOTIC ANALGESIC DRUGS WITH DIFFERENT AGONIST AND ANTAGONIST PROPERTIES [J].

MAGNAN, J ;

PATERSON, SJ ;

TAVANI, A ;

KOSTERLITZ, HW .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 319 (03) :197-205

[6] RABBIT VAS-DEFERENS - A SPECIFIC BIOASSAY FOR OPIOID KAPPA-RECEPTOR AGONISTS [J].

OKA, T ;

NEGISHI, K ;

SUDA, M ;

MATSUMIYA, T ;

INAZU, T ;

UEKI, M .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 73 (2-3) :235-236

[7]

SIMON EJ, 1975, J PHARMACOL EXP THER, V192, P531

[8]

SIMON EJ, 1984, FED P, V43, pP542

[9] THE OPIOID K-SELECTIVE COMPOUND U-50,488H DOES NOT INHIBIT INTESTINAL PROPULSION IN RATS [J].

TAVANI, A ;

GAMBINO, MC ;

PETRILLO, P .

JOURNAL OF PHARMACY AND PHARMACOLOGY, 1984, 36 (05) :343-344

[10]

WARD SJ, 1983, J PHARMACOL EXP THER, V224, P359

← 1 2 →