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Challenges in beta(3)-adrenoceptor agonist drug development
被引:95
作者
:
Arch, Jonathan R. S.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Buckingham, Clore Lab, Hunter St, Buckingham MK18 1EG, England
Univ Buckingham, Clore Lab, Hunter St, Buckingham MK18 1EG, England
Arch, Jonathan R. S.
[
1
]
机构
:
[1]
Univ Buckingham, Clore Lab, Hunter St, Buckingham MK18 1EG, England
来源
:
THERAPEUTIC ADVANCES IN ENDOCRINOLOGY AND METABOLISM
|
2011年
/ 2卷
/ 02期
关键词
:
D O I
:
10.1177/2042018811398517
中图分类号
:
R5 [内科学];
学科分类号
:
1002 ;
100201 ;
摘要
:
引用
收藏
页码:59 / 64
页数:6
相关论文
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[51]
Acute effect of L-796568, a novel β3-adrenergic receptor agonist, on energy expenditure in obese men
[J].
van Baak, MA
论文数:
0
引用数:
0
h-index:
0
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Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
van Baak, MA
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0
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0
h-index:
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Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Hul, GBJ
;
Toubro, S
论文数:
0
引用数:
0
h-index:
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Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Toubro, S
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Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Astrup, A
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0
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0
h-index:
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Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Gottesdiener, KM
;
DeSmet, M
论文数:
0
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0
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Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
DeSmet, M
;
Saris, WHM
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Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Saris, WHM
.
CLINICAL PHARMACOLOGY & THERAPEUTICS,
2002,
71
(04)
:272
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[52]
Chronic treatment with BRL 35135 potentiates the action of insulin on lipid metabolism
[J].
Virtanen, KA
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Dept. Pharmacol. Clin. Pharmacol., University of Turku, FIN-20520 Turku
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Huupponen, R
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EUROPEAN JOURNAL OF PHARMACOLOGY,
1997,
332
(02)
:215
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[53]
Bile acids induce energy expenditure by promoting intracellular thyroid hormone activation
[J].
Watanabe, M
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0
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0
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ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
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Harney, JW
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Ezaki, O
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Auwerx, J
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439
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:484
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[54]
GENETICALLY-OBESE C57BL/6 OB OB MICE RESPOND NORMALLY TO SYMPATHOMIMETIC COMPOUNDS
[J].
WILSON, S
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WILSON, S
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ARCH, JRS
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ARCH, JRS
;
THURLBY, PL
论文数:
0
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THURLBY, PL
.
LIFE SCIENCES,
1984,
35
(12)
:1301
-1309
[55]
SUBSTRATE SUPPLY FOR THERMOGENESIS INDUCED BY THE BETA-ADRENOCEPTOR AGONIST BRL-26830A
[J].
WILSON, S
论文数:
0
引用数:
0
h-index:
0
WILSON, S
;
THURLBY, PL
论文数:
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THURLBY, PL
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ARCH, JRS
论文数:
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h-index:
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ARCH, JRS
.
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY,
1987,
65
(02)
:113
-119
[56]
YEN TT, 1984, INT J OBESITY, V8, P65
←
1
2
3
4
5
6
→
共 56 条
[51]
Acute effect of L-796568, a novel β3-adrenergic receptor agonist, on energy expenditure in obese men
[J].
van Baak, MA
论文数:
0
引用数:
0
h-index:
0
机构:
Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
van Baak, MA
;
Hul, GBJ
论文数:
0
引用数:
0
h-index:
0
机构:
Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Hul, GBJ
;
Toubro, S
论文数:
0
引用数:
0
h-index:
0
机构:
Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Toubro, S
;
Astrup, A
论文数:
0
引用数:
0
h-index:
0
机构:
Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Astrup, A
;
Gottesdiener, KM
论文数:
0
引用数:
0
h-index:
0
机构:
Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Gottesdiener, KM
;
DeSmet, M
论文数:
0
引用数:
0
h-index:
0
机构:
Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
DeSmet, M
;
Saris, WHM
论文数:
0
引用数:
0
h-index:
0
机构:
Maastricht Univ, Dept Human Biol, Nutr & Toxicol Res Inst, NL-6200 MD Maastricht, Netherlands
Saris, WHM
.
CLINICAL PHARMACOLOGY & THERAPEUTICS,
2002,
71
(04)
:272
-279
[52]
Chronic treatment with BRL 35135 potentiates the action of insulin on lipid metabolism
[J].
Virtanen, KA
论文数:
0
引用数:
0
h-index:
0
机构:
Dept. Pharmacol. Clin. Pharmacol., University of Turku, FIN-20520 Turku
Virtanen, KA
;
Rouru, J
论文数:
0
引用数:
0
h-index:
0
机构:
Dept. Pharmacol. Clin. Pharmacol., University of Turku, FIN-20520 Turku
Rouru, J
;
Hanninen, V
论文数:
0
引用数:
0
h-index:
0
机构:
Dept. Pharmacol. Clin. Pharmacol., University of Turku, FIN-20520 Turku
Hanninen, V
;
论文数:
引用数:
h-index:
机构:
Savontaus, E
;
Rouvari, T
论文数:
0
引用数:
0
h-index:
0
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Dept. Pharmacol. Clin. Pharmacol., University of Turku, FIN-20520 Turku
Rouvari, T
;
Teirmaa, T
论文数:
0
引用数:
0
h-index:
0
机构:
Dept. Pharmacol. Clin. Pharmacol., University of Turku, FIN-20520 Turku
Teirmaa, T
;
Koulu, M
论文数:
0
引用数:
0
h-index:
0
机构:
Dept. Pharmacol. Clin. Pharmacol., University of Turku, FIN-20520 Turku
Koulu, M
;
Huupponen, R
论文数:
0
引用数:
0
h-index:
0
机构:
Dept. Pharmacol. Clin. Pharmacol., University of Turku, FIN-20520 Turku
Huupponen, R
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1997,
332
(02)
:215
-218
[53]
Bile acids induce energy expenditure by promoting intracellular thyroid hormone activation
[J].
Watanabe, M
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Watanabe, M
;
Houten, SM
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Houten, SM
;
Mataki, C
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Mataki, C
;
Christoffolete, MA
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Christoffolete, MA
;
Kim, BW
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Kim, BW
;
Sato, H
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Sato, H
;
Messaddeq, N
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Messaddeq, N
;
Harney, JW
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Harney, JW
;
Ezaki, O
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Ezaki, O
;
Kodama, T
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Kodama, T
;
Schoonjans, K
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Schoonjans, K
;
Bianco, AC
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Bianco, AC
;
Auwerx, J
论文数:
0
引用数:
0
h-index:
0
机构:
ULP, CNRS, INSERM, Inst Genet & Biol Mol & Cellulaire, F-67404 Illkirch Graffenstaden, France
Auwerx, J
.
NATURE,
2006,
439
(7075)
:484
-489
[54]
GENETICALLY-OBESE C57BL/6 OB OB MICE RESPOND NORMALLY TO SYMPATHOMIMETIC COMPOUNDS
[J].
WILSON, S
论文数:
0
引用数:
0
h-index:
0
WILSON, S
;
ARCH, JRS
论文数:
0
引用数:
0
h-index:
0
ARCH, JRS
;
THURLBY, PL
论文数:
0
引用数:
0
h-index:
0
THURLBY, PL
.
LIFE SCIENCES,
1984,
35
(12)
:1301
-1309
[55]
SUBSTRATE SUPPLY FOR THERMOGENESIS INDUCED BY THE BETA-ADRENOCEPTOR AGONIST BRL-26830A
[J].
WILSON, S
论文数:
0
引用数:
0
h-index:
0
WILSON, S
;
THURLBY, PL
论文数:
0
引用数:
0
h-index:
0
THURLBY, PL
;
ARCH, JRS
论文数:
0
引用数:
0
h-index:
0
ARCH, JRS
.
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY,
1987,
65
(02)
:113
-119
[56]
YEN TT, 1984, INT J OBESITY, V8, P65
←
1
2
3
4
5
6
→