7-ALPHA-SUBSTITUTED DERIVATIVES OF ANDROSTENEDIONE AS INHIBITORS OF ESTROGEN BIOSYNTHESIS

被引：34

作者：

DARBY, MV ^{[1
]}

LOVETT, JA ^{[1
]}

BRUEGGEMEIER, RW ^{[1
]}

GROZIAK, MP ^{[1
]}

COUNSELL, RE ^{[1
]}

机构：

[1] UNIV MICHIGAN,INTERDEPT PROGRAM MED CHEM,ANN ARBOR,MI 48109

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 06期

关键词：

D O I：

10.1021/jm00383a019

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：803 / 807

页数：5

共 27 条

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[4] EFFECT OF AN AROMATASE INHIBITOR, 1,4,6-ANDROSTATRIENE-3,17-DIONE, ON 7,12-DIMETHYLBENZ (A) ANTHRACENE-INDUCED MAMMARY-TUMORS IN THE RAT AND ITS MECHANISM OF ACTION INVIVO [J].

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[5]

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[6]

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[7]

BRUEGGEMEIER RW, 1982, CANCER RES, V42, P3334

[8] SYNTHESIS AND BIOCHEMICAL EVALUATION OF INHIBITORS OF ESTROGEN BIOSYNTHESIS [J].

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FLOYD, EE ;

COUNSELL, RE .

JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (10) :1007-1011

[9]

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[10]

CAMPBELL MM, 1979, TETRAHEDRON LETT, P2455

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