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COMPARISON OF 2 PENICILLAMINE-CONTAINING ENKEPHALINS - MU, NOT DELTA, ACTIVITY PRODUCES ANALGESIA
被引:12
作者
:
LEANDER, JD
论文数:
0
引用数:
0
h-index:
0
LEANDER, JD
GESELLCHEN, PD
论文数:
0
引用数:
0
h-index:
0
GESELLCHEN, PD
MENDELSOHN, LG
论文数:
0
引用数:
0
h-index:
0
MENDELSOHN, LG
机构
:
来源
:
NEUROPEPTIDES
|
1986年
/ 8卷
/ 02期
关键词
:
D O I
:
10.1016/0143-4179(86)90038-7
中图分类号
:
R5 [内科学];
学科分类号
:
1002 ;
100201 ;
摘要
:
引用
收藏
页码:119 / 125
页数:7
相关论文
共 17 条
[1]
THE MU-RATHER THAN THE DELTA-SUBTYPE OF OPIOID RECEPTORS APPEARS TO BE INVOLVED IN ENKEPHALIN-INDUCED ANALGESIA
[J].
CHAILLET, P
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
CHAILLET, P
;
COULAUD, A
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
COULAUD, A
;
ZAJAC, JM
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
ZAJAC, JM
;
FOURNIEZALUSKI, MC
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
FOURNIEZALUSKI, MC
;
COSTENTIN, J
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
COSTENTIN, J
;
ROQUES, BP
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
ROQUES, BP
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1984,
101
(1-2)
:83
-90
[2]
ABDOMINAL CONSTRICTION RESPONSE AND ITS SUPPRESSION BY ANALGESIC DRUGS IN MOUSE
[J].
COLLIER, HOJ
论文数:
0
引用数:
0
h-index:
0
COLLIER, HOJ
;
DINNEEN, LC
论文数:
0
引用数:
0
h-index:
0
DINNEEN, LC
;
JOHNSON, CA
论文数:
0
引用数:
0
h-index:
0
JOHNSON, CA
;
SCHNEIDER, C
论文数:
0
引用数:
0
h-index:
0
SCHNEIDER, C
.
BRITISH JOURNAL OF PHARMACOLOGY,
1968,
32
(02)
:295
-+
[3]
SELECTIVITIES OF OPIOID PEPTIDE ANALOGS AS AGONISTS AND ANTAGONISTS AT THE DELTA-RECEPTOR
[J].
CORBETT, AD
论文数:
0
引用数:
0
h-index:
0
CORBETT, AD
;
GILLAN, MGC
论文数:
0
引用数:
0
h-index:
0
GILLAN, MGC
;
KOSTERLITZ, HW
论文数:
0
引用数:
0
h-index:
0
KOSTERLITZ, HW
;
MCKNIGHT, AT
论文数:
0
引用数:
0
h-index:
0
MCKNIGHT, AT
;
PATERSON, SJ
论文数:
0
引用数:
0
h-index:
0
PATERSON, SJ
;
ROBSON, LE
论文数:
0
引用数:
0
h-index:
0
ROBSON, LE
.
BRITISH JOURNAL OF PHARMACOLOGY,
1984,
83
(01)
:271
-279
[4]
ICI-174864 - A HIGHLY SELECTIVE ANTAGONIST FOR THE OPIOID DELTA-RECEPTOR
[J].
COTTON, R
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
COTTON, R
;
GILES, MG
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
GILES, MG
;
MILLER, L
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
MILLER, L
;
SHAW, JS
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
SHAW, JS
;
TIMMS, D
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
TIMMS, D
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1984,
97
(3-4)
:331
-332
[5]
EVIDENCE OF THE PREFERENTIAL INVOLVEMENT OF MU-RECEPTORS IN ANALGESIA USING ENKEPHALINS HIGHLY SELECTIVE FOR PERIPHERAL MU-RECEPTOR OR DELTA-RECEPTOR
[J].
GACEL, G
论文数:
0
引用数:
0
h-index:
0
机构:
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
GACEL, G
;
FOURNIEZALUSKI, MC
论文数:
0
引用数:
0
h-index:
0
机构:
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FOURNIEZALUSKI, MC
;
FELLION, E
论文数:
0
引用数:
0
h-index:
0
机构:
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FELLION, E
;
ROQUES, BP
论文数:
0
引用数:
0
h-index:
0
机构:
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
ROQUES, BP
.
JOURNAL OF MEDICINAL CHEMISTRY,
1981,
24
(10)
:1119
-1124
[6]
GALLIGAN GJ, 1984, J PHARM EXP THER, V229, P341
[7]
SPECTRUM OF THE MU-BINDING, DELTA-BINDING AND KAPPA-BINDING SITES IN HOMOGENATES OF RAT-BRAIN
[J].
GILLAN, MGC
论文数:
0
引用数:
0
h-index:
0
GILLAN, MGC
;
KOSTERLITZ, HW
论文数:
0
引用数:
0
h-index:
0
KOSTERLITZ, HW
.
BRITISH JOURNAL OF PHARMACOLOGY,
1982,
77
(03)
:461
-468
[8]
MULTIPLE OPIOID RECEPTORS - CRITERIA FOR IDENTIFICATION AND CLASSIFICATION
[J].
GOLDSTEIN, A
论文数:
0
引用数:
0
h-index:
0
机构:
STANFORD UNIV,PALO ALTO,CA 94304
STANFORD UNIV,PALO ALTO,CA 94304
GOLDSTEIN, A
;
JAMES, IF
论文数:
0
引用数:
0
h-index:
0
机构:
STANFORD UNIV,PALO ALTO,CA 94304
STANFORD UNIV,PALO ALTO,CA 94304
JAMES, IF
.
TRENDS IN PHARMACOLOGICAL SCIENCES,
1984,
5
(12)
:503
-505
[9]
NOVEL PHENYLPIPERIDINE OPIOID ANTAGONISTS AND PARTIAL AGONISTS - EFFECTS ON FLUID CONSUMPTION
[J].
LEANDER, JD
论文数:
0
引用数:
0
h-index:
0
LEANDER, JD
;
HART, JC
论文数:
0
引用数:
0
h-index:
0
HART, JC
;
LOCHNER, MA
论文数:
0
引用数:
0
h-index:
0
LOCHNER, MA
;
HYNES, MD
论文数:
0
引用数:
0
h-index:
0
HYNES, MD
;
ZIMMERMAN, DM
论文数:
0
引用数:
0
h-index:
0
ZIMMERMAN, DM
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1982,
81
(02)
:185
-192
[10]
THE BINDING SPECTRUM OF NARCOTIC ANALGESIC DRUGS WITH DIFFERENT AGONIST AND ANTAGONIST PROPERTIES
[J].
MAGNAN, J
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
MAGNAN, J
;
PATERSON, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
PATERSON, SJ
;
TAVANI, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
TAVANI, A
;
KOSTERLITZ, HW
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
KOSTERLITZ, HW
.
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY,
1982,
319
(03)
:197
-205
←
1
2
→
共 17 条
[1]
THE MU-RATHER THAN THE DELTA-SUBTYPE OF OPIOID RECEPTORS APPEARS TO BE INVOLVED IN ENKEPHALIN-INDUCED ANALGESIA
[J].
CHAILLET, P
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
CHAILLET, P
;
COULAUD, A
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
COULAUD, A
;
ZAJAC, JM
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
ZAJAC, JM
;
FOURNIEZALUSKI, MC
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
FOURNIEZALUSKI, MC
;
COSTENTIN, J
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
COSTENTIN, J
;
ROQUES, BP
论文数:
0
引用数:
0
h-index:
0
机构:
UER SCI PHARMACEUT & BIOL, INSERM 266, 4 AVE OBSERV, F-75006 PARIS, FRANCE
ROQUES, BP
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1984,
101
(1-2)
:83
-90
[2]
ABDOMINAL CONSTRICTION RESPONSE AND ITS SUPPRESSION BY ANALGESIC DRUGS IN MOUSE
[J].
COLLIER, HOJ
论文数:
0
引用数:
0
h-index:
0
COLLIER, HOJ
;
DINNEEN, LC
论文数:
0
引用数:
0
h-index:
0
DINNEEN, LC
;
JOHNSON, CA
论文数:
0
引用数:
0
h-index:
0
JOHNSON, CA
;
SCHNEIDER, C
论文数:
0
引用数:
0
h-index:
0
SCHNEIDER, C
.
BRITISH JOURNAL OF PHARMACOLOGY,
1968,
32
(02)
:295
-+
[3]
SELECTIVITIES OF OPIOID PEPTIDE ANALOGS AS AGONISTS AND ANTAGONISTS AT THE DELTA-RECEPTOR
[J].
CORBETT, AD
论文数:
0
引用数:
0
h-index:
0
CORBETT, AD
;
GILLAN, MGC
论文数:
0
引用数:
0
h-index:
0
GILLAN, MGC
;
KOSTERLITZ, HW
论文数:
0
引用数:
0
h-index:
0
KOSTERLITZ, HW
;
MCKNIGHT, AT
论文数:
0
引用数:
0
h-index:
0
MCKNIGHT, AT
;
PATERSON, SJ
论文数:
0
引用数:
0
h-index:
0
PATERSON, SJ
;
ROBSON, LE
论文数:
0
引用数:
0
h-index:
0
ROBSON, LE
.
BRITISH JOURNAL OF PHARMACOLOGY,
1984,
83
(01)
:271
-279
[4]
ICI-174864 - A HIGHLY SELECTIVE ANTAGONIST FOR THE OPIOID DELTA-RECEPTOR
[J].
COTTON, R
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
COTTON, R
;
GILES, MG
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
GILES, MG
;
MILLER, L
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
MILLER, L
;
SHAW, JS
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
SHAW, JS
;
TIMMS, D
论文数:
0
引用数:
0
h-index:
0
机构:
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI LTD,DIV PHARMACEUT,DEPT BIOSCI,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
TIMMS, D
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1984,
97
(3-4)
:331
-332
[5]
EVIDENCE OF THE PREFERENTIAL INVOLVEMENT OF MU-RECEPTORS IN ANALGESIA USING ENKEPHALINS HIGHLY SELECTIVE FOR PERIPHERAL MU-RECEPTOR OR DELTA-RECEPTOR
[J].
GACEL, G
论文数:
0
引用数:
0
h-index:
0
机构:
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
GACEL, G
;
FOURNIEZALUSKI, MC
论文数:
0
引用数:
0
h-index:
0
机构:
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FOURNIEZALUSKI, MC
;
FELLION, E
论文数:
0
引用数:
0
h-index:
0
机构:
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FELLION, E
;
ROQUES, BP
论文数:
0
引用数:
0
h-index:
0
机构:
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
FAC PHARM PARIS, DEPT CHIM ORGAN, CNRS, ERA 613, F-75270 PARIS 06, FRANCE
ROQUES, BP
.
JOURNAL OF MEDICINAL CHEMISTRY,
1981,
24
(10)
:1119
-1124
[6]
GALLIGAN GJ, 1984, J PHARM EXP THER, V229, P341
[7]
SPECTRUM OF THE MU-BINDING, DELTA-BINDING AND KAPPA-BINDING SITES IN HOMOGENATES OF RAT-BRAIN
[J].
GILLAN, MGC
论文数:
0
引用数:
0
h-index:
0
GILLAN, MGC
;
KOSTERLITZ, HW
论文数:
0
引用数:
0
h-index:
0
KOSTERLITZ, HW
.
BRITISH JOURNAL OF PHARMACOLOGY,
1982,
77
(03)
:461
-468
[8]
MULTIPLE OPIOID RECEPTORS - CRITERIA FOR IDENTIFICATION AND CLASSIFICATION
[J].
GOLDSTEIN, A
论文数:
0
引用数:
0
h-index:
0
机构:
STANFORD UNIV,PALO ALTO,CA 94304
STANFORD UNIV,PALO ALTO,CA 94304
GOLDSTEIN, A
;
JAMES, IF
论文数:
0
引用数:
0
h-index:
0
机构:
STANFORD UNIV,PALO ALTO,CA 94304
STANFORD UNIV,PALO ALTO,CA 94304
JAMES, IF
.
TRENDS IN PHARMACOLOGICAL SCIENCES,
1984,
5
(12)
:503
-505
[9]
NOVEL PHENYLPIPERIDINE OPIOID ANTAGONISTS AND PARTIAL AGONISTS - EFFECTS ON FLUID CONSUMPTION
[J].
LEANDER, JD
论文数:
0
引用数:
0
h-index:
0
LEANDER, JD
;
HART, JC
论文数:
0
引用数:
0
h-index:
0
HART, JC
;
LOCHNER, MA
论文数:
0
引用数:
0
h-index:
0
LOCHNER, MA
;
HYNES, MD
论文数:
0
引用数:
0
h-index:
0
HYNES, MD
;
ZIMMERMAN, DM
论文数:
0
引用数:
0
h-index:
0
ZIMMERMAN, DM
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1982,
81
(02)
:185
-192
[10]
THE BINDING SPECTRUM OF NARCOTIC ANALGESIC DRUGS WITH DIFFERENT AGONIST AND ANTAGONIST PROPERTIES
[J].
MAGNAN, J
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
MAGNAN, J
;
PATERSON, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
PATERSON, SJ
;
TAVANI, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
TAVANI, A
;
KOSTERLITZ, HW
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
UNIV ABERDEEN, MARISCHAL COLL, RES ADDICT DRUGS UNIT, ABERDEEN AB9 1AS, SCOTLAND
KOSTERLITZ, HW
.
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY,
1982,
319
(03)
:197
-205
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