COMPARISON OF 2 PENICILLAMINE-CONTAINING ENKEPHALINS - MU, NOT DELTA, ACTIVITY PRODUCES ANALGESIA

被引:12
作者
LEANDER, JD
GESELLCHEN, PD
MENDELSOHN, LG
机构
关键词
D O I
10.1016/0143-4179(86)90038-7
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
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页码:119 / 125
页数:7
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共 17 条
[1]   THE MU-RATHER THAN THE DELTA-SUBTYPE OF OPIOID RECEPTORS APPEARS TO BE INVOLVED IN ENKEPHALIN-INDUCED ANALGESIA [J].
CHAILLET, P ;
COULAUD, A ;
ZAJAC, JM ;
FOURNIEZALUSKI, MC ;
COSTENTIN, J ;
ROQUES, BP .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 101 (1-2) :83-90
[2]   ABDOMINAL CONSTRICTION RESPONSE AND ITS SUPPRESSION BY ANALGESIC DRUGS IN MOUSE [J].
COLLIER, HOJ ;
DINNEEN, LC ;
JOHNSON, CA ;
SCHNEIDER, C .
BRITISH JOURNAL OF PHARMACOLOGY, 1968, 32 (02) :295-+
[3]   SELECTIVITIES OF OPIOID PEPTIDE ANALOGS AS AGONISTS AND ANTAGONISTS AT THE DELTA-RECEPTOR [J].
CORBETT, AD ;
GILLAN, MGC ;
KOSTERLITZ, HW ;
MCKNIGHT, AT ;
PATERSON, SJ ;
ROBSON, LE .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 83 (01) :271-279
[4]   ICI-174864 - A HIGHLY SELECTIVE ANTAGONIST FOR THE OPIOID DELTA-RECEPTOR [J].
COTTON, R ;
GILES, MG ;
MILLER, L ;
SHAW, JS ;
TIMMS, D .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 97 (3-4) :331-332
[5]   EVIDENCE OF THE PREFERENTIAL INVOLVEMENT OF MU-RECEPTORS IN ANALGESIA USING ENKEPHALINS HIGHLY SELECTIVE FOR PERIPHERAL MU-RECEPTOR OR DELTA-RECEPTOR [J].
GACEL, G ;
FOURNIEZALUSKI, MC ;
FELLION, E ;
ROQUES, BP .
JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (10) :1119-1124
[6]  
GALLIGAN GJ, 1984, J PHARM EXP THER, V229, P341
[7]   SPECTRUM OF THE MU-BINDING, DELTA-BINDING AND KAPPA-BINDING SITES IN HOMOGENATES OF RAT-BRAIN [J].
GILLAN, MGC ;
KOSTERLITZ, HW .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 77 (03) :461-468
[8]   MULTIPLE OPIOID RECEPTORS - CRITERIA FOR IDENTIFICATION AND CLASSIFICATION [J].
GOLDSTEIN, A ;
JAMES, IF .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1984, 5 (12) :503-505
[9]   NOVEL PHENYLPIPERIDINE OPIOID ANTAGONISTS AND PARTIAL AGONISTS - EFFECTS ON FLUID CONSUMPTION [J].
LEANDER, JD ;
HART, JC ;
LOCHNER, MA ;
HYNES, MD ;
ZIMMERMAN, DM .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 81 (02) :185-192
[10]   THE BINDING SPECTRUM OF NARCOTIC ANALGESIC DRUGS WITH DIFFERENT AGONIST AND ANTAGONIST PROPERTIES [J].
MAGNAN, J ;
PATERSON, SJ ;
TAVANI, A ;
KOSTERLITZ, HW .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 319 (03) :197-205