A SELECTIVE IMIDAZOBENZODIAZEPINE ANTAGONIST OF ETHANOL IN THE RAT

被引:522
作者
SUZDAK, PD
GLOWA, JR
CRAWLEY, JN
SCHWARTZ, RD
SKOLNICK, P
PAUL, SM
机构
[1] NIMH,CLIN NEUROSCI BRANCH,MOLEC PHARMACOL & PRECLIN STUDIES SECT,BLDG 10,ROOM 4N214,BETHESDA,MD 20892
[2] NIDDKD,BIOORGAN CHEM LAB,NEUROBIOL SECT,BETHESDA,MD 20892
关键词
D O I
10.1126/science.3022383
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:1243 / 1247
页数:5
相关论文
共 56 条
[1]  
[Anonymous], ALCOHOL BIOL MEMBRAN
[2]  
BONETTI E P, 1985, British Journal of Pharmacology, V86, p463P
[3]   LIGANDS FOR BENZODIAZEPINE RECEPTORS WITH POSITIVE AND NEGATIVE EFFICACY [J].
BRAESTRUP, C ;
HONORE, T ;
NIELSEN, M ;
PETERSEN, EN ;
JENSEN, LH .
BIOCHEMICAL PHARMACOLOGY, 1984, 33 (06) :859-862
[4]   ETHANOL IN LOW-DOSES AUGMENTS CALCIUM-MEDIATED MECHANISMS MEASURED INTRACELLULARLY IN HIPPOCAMPAL-NEURONS [J].
CARLEN, PL ;
GUREVICH, N ;
DURAND, D .
SCIENCE, 1982, 215 (4530) :306-309
[5]  
CHIN JH, 1977, MOL PHARMACOL, V13, P435
[6]  
COLE JO, 1975, AM HDB PSYCHIATRY, P427
[7]   NEW CONCEPTS ON MECHANISM OF ACTION OF BENZODIAZEPINES [J].
COSTA, E ;
GUIDOTTI, A ;
MAO, CC ;
SURIA, A .
LIFE SCIENCES, 1975, 17 (02) :167-185
[8]   ABSENCE OF INTRINSIC ANTAGONIST ACTIONS OF BENZODIAZEPINE ANTAGONISTS ON AN EXPLORATORY MODEL OF ANXIETY IN THE MOUSE [J].
CRAWLEY, JN ;
SKOLNICK, P ;
PAUL, SM .
NEUROPHARMACOLOGY, 1984, 23 (05) :531-537
[9]   CGS-8216 - RECEPTOR-BINDING CHARACTERISTICS OF A POTENT BENZODIAZEPINE ANTAGONIST [J].
CZERNIK, AJ ;
PETRACK, B ;
KALINSKY, HJ ;
PSYCHOYOS, S ;
CASH, WD ;
TSAI, C ;
RINEHART, RK ;
GRANAT, FR ;
LOVELL, RA ;
BRUNDISH, DE ;
WADE, R .
LIFE SCIENCES, 1982, 30 (04) :363-372
[10]   ALCOHOL AND PRESYNAPTIC INHIBITION IN AN ISOLATED SPINAL-CORD PREPARATION [J].
DAVIDOFF, RA .
ARCHIVES OF NEUROLOGY, 1973, 28 (01) :60-63