A SELECTIVE IMIDAZOBENZODIAZEPINE ANTAGONIST OF ETHANOL IN THE RAT

被引:522
作者
SUZDAK, PD
GLOWA, JR
CRAWLEY, JN
SCHWARTZ, RD
SKOLNICK, P
PAUL, SM
机构
[1] NIMH,CLIN NEUROSCI BRANCH,MOLEC PHARMACOL & PRECLIN STUDIES SECT,BLDG 10,ROOM 4N214,BETHESDA,MD 20892
[2] NIDDKD,BIOORGAN CHEM LAB,NEUROBIOL SECT,BETHESDA,MD 20892
关键词
D O I
10.1126/science.3022383
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:1243 / 1247
页数:5
相关论文
共 56 条
[31]   LOW-DOSES OF ETHANOL INHIBIT THE FIRING OF NEURONS IN THE SUBSTANTIA-NIGRA, PARS RETICULATA - A GABAERGIC EFFECT [J].
MEREU, G ;
GESSA, GL .
BRAIN RESEARCH, 1985, 360 (1-2) :325-330
[32]   ALCOHOL EFFECTS ON SYNAPTIC MEMBRANE CALCIUM-ION FLUXES [J].
MICHAELIS, ML ;
MICHAELIS, EK ;
TEHAN, T .
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1983, 18 :19-23
[33]   ALCOHOL AND LOCAL-ANESTHETIC EFFECTS ON NA+- DEPENDENT CA-2+ FLUXES IN BRAIN SYNAPTIC MEMBRANE-VESICLES [J].
MICHAELIS, ML ;
MICHAELIS, EK .
BIOCHEMICAL PHARMACOLOGY, 1983, 32 (06) :963-969
[34]   PHOTOAFFINITY-LABELING OF BENZODIAZEPINE RECEPTORS WITH A PARTIAL INVERSE AGONIST [J].
MOHLER, H ;
SIEGHART, W ;
RICHARDS, JG ;
HUNKELER, W .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 102 (01) :191-192
[35]   ETHANOL INHIBITS VERATRIDINE-STIMULATED SODIUM UPTAKE IN SYNAPTOSOMES [J].
MULLIN, MJ ;
HUNT, WA .
LIFE SCIENCES, 1984, 34 (03) :287-292
[36]   ETHANOL SPECIFICALLY POTENTIATES GABA-MEDIATED NEUROTRANSMISSION IN FELINE CEREBRAL-CORTEX [J].
NESTOROS, JN .
SCIENCE, 1980, 209 (4457) :708-710
[37]   PROLONGATION OF HIPPOCAMPAL INHIBITORY POSTSYNAPTIC POTENTIALS BY BARBITURATES [J].
NICOLL, RA ;
ECCLES, JC ;
OSHIMA, T ;
RUBIA, F .
NATURE, 1975, 258 (5536) :625-627
[38]   GABA-BENZODIAZEPINE-BARBITURATE RECEPTOR INTERACTIONS [J].
OLSEN, RW .
JOURNAL OF NEUROCHEMISTRY, 1981, 37 (01) :1-13
[39]   DRUG-INTERACTIONS AT THE GABA RECEPTOR-IONOPHORE COMPLEX [J].
OLSEN, RW .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1982, 22 :245-277
[40]   GABA RECEPTOR MEDIATED CHLORIDE TRANSPORT IN A CELL-FREE MEMBRANE PREPARATION FROM BRAIN [J].
PAUL, SM ;
SCHWARTZ, RD ;
CREVELING, CR ;
HOLLINGSWORTH, EB ;
DALY, JW ;
SKOLNICK, P .
SCIENCE, 1986, 233 (4760) :228-229