SYNTHESIS OF NOVEL 2-SUBSTITUTED-5-OXYCOUMARANS VIA A DIRECT ROUTE TO 2,3-DIHYDRO-5-HYDROXY-2-BENZOFURANACETIC ACIDS

被引：17

作者：

CECCARELLI, S ^{[1
]}

DEVELLIS, P ^{[1
]}

SCURI, R ^{[1
]}

ZANARELLA, S ^{[1
]}

BRUFANI, M ^{[1
]}

机构：

[1] UNIV ROMA LA SAPIENZA, DIPARTIMENTO SCI BIOCHIM A ROSSI FANELLI, I-00185 ROME, ITALY

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1993年 / 30卷 / 03期

关键词：

D O I：

10.1002/jhet.5570300318

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A number of novel 2-substituted 2,3-dihydro-5-benzofuranols optionally protected on 5-OH group have been prepared via a simple two step route to racemic 2,3-dihydro-5-hydroxy-2-benzofuranacetic acids from hydroquinones and 4-bromocrotonates.

引用

页码：679 / 690

页数：12

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