COMPARISON BETWEEN INVIVO AND INVITRO TISSUE-TO-PLASMA UNBOUND CONCENTRATION RATIOS (KP,F) OF QUINIDINE IN RATS

被引:33
作者
HARASHIMA, H [1 ]
SUGIYAMA, Y [1 ]
SAWADA, Y [1 ]
IGA, T [1 ]
机构
[1] UNIV TOKYO,FAC PHARMACEUT SCI,BUNKYO KU,TOKYO 113,JAPAN
关键词
D O I
10.1111/j.2042-7158.1984.tb04390.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:340 / 342
页数:3
相关论文
共 20 条
[1]  
BIARCHETTI G, 1980, J PHARM EXP THER, V214, P682
[2]  
BICKEL MH, 1975, LIVER, P130
[3]   ESTIMATION OF TISSUE-TO-PLASMA PARTITION-COEFFICIENTS USED IN PHYSIOLOGICAL PHARMACOKINETIC MODELS [J].
CHEN, HSG ;
GROSS, JF .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1979, 7 (01) :117-125
[4]   QUANTITATIVE DETERMINATION OF QUINIDINE IN PLASMA [J].
CRAMER, G ;
ISAKSSON, B .
SCANDINAVIAN JOURNAL OF CLINICAL & LABORATORY INVESTIGATION, 1963, 15 (05) :553-&
[5]   MEMBRANE LIPIDS AS INTRACELLULAR BINDERS OF CHLORPROMAZINE AND RELATED DRUGS [J].
DIFRANCESCO, C ;
BICKEL, MH .
CHEMICO-BIOLOGICAL INTERACTIONS, 1977, 16 (03) :335-346
[6]  
EILING TE, 1975, DRUG METAB DISPOS, V3, P389
[7]  
FICHTL B, 1980, J PHARMACOL EXP THER, V215, P248
[8]  
HARASHIMA H, 1983, 102TH ANN M JAP PHAR
[9]   REVIEW OF THE APPLICATIONS OF PHYSIOLOGICALLY BASED PHARMACOKINETIC MODELING [J].
HIMMELSTEIN, KJ ;
LUTZ, RJ .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1979, 7 (02) :127-145
[10]   5-HYDROXYTRYPTAMINE BINDING TO BUTANOL EXTRACTS FROM MYELIN FRAGMENTS [J].
ISHITANI, R ;
MIYAKAWA, A ;
SAITO, R ;
IWAMOTO, T .
EXPERIENTIA, 1977, 33 (07) :932-933