PHOTOAFFINITY-LABELING OF THE BENZODIAZEPINE RECEPTOR COMPROMISES THE RECOGNITION SITE BUT NOT ITS EFFECTOR MECHANISM

被引：9

作者：

BROWN, CL ^{[1
]}

MARTIN, IL ^{[1
]}

机构：

[1] MED SCH CAMBRIDGE,MRC CTR,NEUROCHEM PHARMACOL UNIT,CAMBRIDGE CB2 2QH,ENGLAND

来源：

JOURNAL OF NEUROCHEMISTRY | 1984年 / 43卷 / 01期

关键词：

D O I：

10.1111/j.1471-4159.1984.tb06707.x

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：272 / 273

页数：2

共 15 条

[1]

BROWN C L, 1982, British Journal of Pharmacology, V77, p312P

[2] PHOTOAFFINITY-LABELING OF THE BENZODIAZEPINE RECEPTOR CANNOT BE USED TO PREDICT LIGAND EFFICACY [J].

BROWN, CL ;

MARTIN, IL .

NEUROSCIENCE LETTERS, 1983, 35 (01) :37-40

[3]

COSTA T, 1981, MOL PHARMACOL, V20, P470

[4] IS THE BENZODIAZEPINE RECEPTOR COUPLED TO A CHLORIDE ANION CHANNEL [J].

COSTA, T ;

RODBARD, D ;

PERT, CB .

NATURE, 1979, 277 (5694) :315-317

[5]

DOBLE A, 1982, British Journal of Pharmacology, V76, p238P

[6] BINDING-ENERGY AND THE ACTIVATION OF HORMONE RECEPTORS [J].

FRANKLIN, TJ .

BIOCHEMICAL PHARMACOLOGY, 1980, 29 (06) :853-856

[7] STIMULATION OF BENZODIAZEPINE RECEPTOR-BINDING BY GAMMA-AMINOBUTYRIC ACID [J].

KAROBATH, M ;

SPERK, G .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1979, 76 (02) :1004-1006

[8] DISTINCTION OF BENZODIAZEPINE AGONISTS FROM ANTAGONISTS BY PHOTOAFFINITY-LABELING OF BENZODIAZEPINE RECEPTORS INVITRO [J].

KAROBATH, M ;

SUPAVILAI, P .

NEUROSCIENCE LETTERS, 1982, 31 (01) :65-69

[9] FACILITATION OF BENZODIAZEPINE BINDING BY SODIUM-CHLORIDE AND GABA [J].

MARTIN, IL ;

CANDY, JM .

NEUROPHARMACOLOGY, 1978, 17 (11) :993-998

[10] AGONIST AND ANTAGONIST BENZODIAZEPINE RECEPTOR INTERACTION INVITRO [J].

MOHLER, H ;

RICHARDS, JG .

NATURE, 1981, 294 (5843) :763-765

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