STRUCTURE ACTIVITY RELATIONSHIPS AMONG BENEXTRAMINE-RELATED TETRAAMINE DISULFIDES AT PERIPHERAL ALPHA-ADRENORECEPTORS

被引：8

作者：

ANGELI, P ^{[1
]}

BRASILI, L ^{[1
]}

BRANCIA, E ^{[1
]}

GIARDINA, D ^{[1
]}

QUAGLIA, W ^{[1
]}

MELCHIORRE, C ^{[1
]}

机构：

[1] UNIV CAMERINO,DEPT CHEM SCI,I-62032 CAMERINO,ITALY

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 11期

关键词：

D O I：

10.1021/jm00149a017

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1643 / 1647

页数：5

共 22 条

[1] SYNTHESES RELATED TO ETIOJERVANE .1. SYNTHESIS OF 1,8-DIMETHYL-7-METHOXY-1,2,3,4,4A,9A-HEXAHYDROFLUORENONE-2-CARBOXYLIC ACID [J].

BARNES, RA ;

GERBER, NN .

JOURNAL OF ORGANIC CHEMISTRY, 1961, 26 (11) :4540-&

[2] IRREVERSIBLE ALPHA-ADRENOCEPTOR BLOCKING EFFECTS AND REVERSIBLE MUSCARINIC BLOCKING AND NICOTINIC BLOCKING EFFECTS OF TETRAMINE DISULFIDES ON THE HEART [J].

BENFEY, BG ;

BELLEAU, B ;

BRASILI, L ;

GIANNELLA, M ;

MELCHIORRE, C .

CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1980, 58 (12) :1477-1483

[3] INHIBITION OF THE CARDIAC INOTROPIC EFFECT OF PHENYLEPHRINE BY A TETRAMINE DISULFIDE WITH IRREVERSIBLE ALPHA-ADRENOCEPTOR BLOCKING ACTIVITY [J].

BENFEY, BG ;

YONG, MS ;

BELLEAU, B ;

MELCHIORRE, C .

CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1979, 57 (05) :510-516

[4] REACTIVATION BY CYSTEAMINE OF VASCULAR ALPHA-ADRENOCEPTORS BLOCKED BY THE TETRAMINE DISULFIDE BENEXTRAMINE AND INTERACTION OF BENEXTRAMINE WITH PHENOXYBENZAMINE [J].

BRASILI, L ;

MELCHIORRE, C ;

BELLEAU, B ;

BENFEY, BG .

CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1980, 58 (12) :1490-1493

[5] N,N''-(DITHIO-2,1-ETHANEDIYL)BIS(N'-(PYRROL-2-YLMETHYL)-1,6-HEXANEDIAMINE)(PYREXTRAMINE), A NEW IRREVERSIBLE ALPHA-1-ADRENORECEPTOR BLOCKING-AGENT OF THE TETRAMINE DISULFIDE CLASS [J].

BRASILI, L ;

ANGELI, P ;

BRANCIA, E ;

MELCHIORRE, C .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 103 (1-2) :181-184

[6]

BRAZENOR RM, 1981, J PHARMACOL EXP THER, V218, P530

[7]

CANTACUZENE D, 1979, SCIENCE WASHINGTON, P1217

[8] DEMONSTRATION OF ALPHA-1S-ADRENOCEPTORS AFTER EXPOSURE OF THE RAT ANOCOCCYGEUS TO BENEXTRAMINE [J].

COATES, J ;

WEETMAN, DF .

BRITISH JOURNAL OF PHARMACOLOGY, 1983, 80 (02) :343-346

[9] UMSETZUNG SCHWEFELHALTIGER BENZALDEHYDE MIT DIAZOMETHAN [J].

EISTERT, B ;

SELZER, H ;

SCHADE, W .

CHEMISCHE BERICHTE-RECUEIL, 1964, 97 (05) :1470-&

[10]

FURCHGOTT RF, 1980, VASCULAR NEUROEFFECT, P245

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