POLYOLS OF A CASCADE TYPE AS A WATER-SOLUBILIZING ELEMENT OF CARBORANE DERIVATIVES FOR BORON NEUTRON-CAPTURE THERAPY

被引：80

作者：

NEMOTO, H ^{[1
]}

WILSON, JG ^{[1
]}

NAKAMURA, H ^{[1
]}

YAMAMOTO, Y ^{[1
]}

机构：

[1] TOHOKU UNIV,FAC SCI,DEPT CHEM,SENDAI,MIYAGI 980,JAPAN

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1992年 / 57卷 / 02期

关键词：

D O I：

10.1021/jo00028a010

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A practical method for the synthesis of polyols of a cascade type, as a water-solubilizing element of carborane derivatives for boron neutron capture therapy (BNCT), was developed. The carborane attached to the tetraol 6a was dissolved in water in a concentration of 5.44 M.

引用

收藏

页码：435 / 435

页数：1

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