ANTICONVULSANT ACTIVITY OF INTRACEREBROVENTRICULARLY ADMINISTERED GLIAL GABA UPTAKE INHIBITORS AND OTHER GABAMIMETICS IN CHEMICAL SEIZURE MODELS

被引:30
作者
GONSALVES, SF
TWITCHELL, B
HARBAUGH, RE
KROGSGAARDLARSEN, P
SCHOUSBOE, A
机构
[1] ROYAL DANISH SCH PHARM,DEPT CHEM BC,PHARMABIOTEC RES CTR,DK-2100 COPENHAGEN,DENMARK
[2] UNIV COPENHAGEN,PANUM INST,DEPT BIOCHEM A,PHARMABIOTEC RES CTR,DK-2200 COPENHAGEN,DENMARK
[3] DARTMOUTH COLL,HITCHCOCK MED CTR,DARTMOUTH MED SCH,DEPT PHARMACOL,HANOVER,NH 03756
关键词
D O I
10.1016/0920-1211(89)90056-9
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
引用
收藏
页码:34 / 41
页数:8
相关论文
共 41 条
[1]   ANTI-CONVULSANT ACTIVITY OF GABA UPTAKE INHIBITORS AND THEIR PRODRUGS FOLLOWING CENTRAL OR SYSTEMIC ADMINISTRATION [J].
CROUCHER, MJ ;
MELDRUM, BS ;
KROGSGAARDLARSEN, P .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 89 (3-4) :217-228
[2]  
CURTIS DR, 1976, EXP BRAIN RES, V25, P413
[3]   THE PERSPECTIVE OF GABA REPLENISHMENT THERAPY IN THE EPILEPSIES - A CRITICAL-EVALUATION OF HOPES AND CONCERNS [J].
FARIELLO, RG ;
TICKU, MK .
LIFE SCIENCES, 1983, 33 (17) :1629-1640
[4]   INFLUENCE OF INHIBITORS OF THE HIGH-AFFINITY GABA UPTAKE ON SEIZURE THRESHOLDS IN MICE [J].
FREY, HH ;
POPP, C ;
LOSCHER, W .
NEUROPHARMACOLOGY, 1979, 18 (07) :581-590
[5]  
GALE K, 1984, NEUROTRANSMITTERS SE, V2, P57
[6]  
HAEFELY W, 1979, A BENZON S, V12, P357
[7]   ANTICONVULSANT ACTIVITY OF THE NIPECOTIC ACID ESTER, (+/-)-META-NITROPHENYL-3-PIPERIDINECARBOXYLATE [J].
HINKO, CN ;
SEIBERT, K ;
CRIDER, AM .
NEUROPHARMACOLOGY, 1984, 23 (09) :1009-1014
[8]   CONVULSANT AND ANTICONVULSANT ACTIONS IN DBA-2 MICE OF COMPOUNDS BLOCKING THE REUPTAKE OF GABA [J].
HORTON, RW ;
COLLINS, JF ;
ANLEZARK, GM ;
MELDRUM, BS .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 59 (1-2) :75-83
[9]   SUBSTANTIA NIGRA - SITE OF ANTICONVULSANT ACTIVITY MEDIATED BY GAMMA-AMINOBUTYRIC ACID [J].
IADAROLA, MJ ;
GALE, K .
SCIENCE, 1982, 218 (4578) :1237-1240
[10]   UPTAKE AND METABOLISM OF GAMMA-AMINOBUTYRIC ACID BY NEURONS AND GLIAL CELLS [J].
IVERSEN, LL ;
KELLY, JS .
BIOCHEMICAL PHARMACOLOGY, 1975, 24 (09) :933-938