TOTAL SYNTHESIS OF (+)-PIPERAZINOMYCIN

被引：56

作者：

BOGER, DL

ZHOU, JC

机构：

[1] Department of Chemistry, The Scripps Research Institute, La Jolla, California 92037

来源：

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY | 1993年 / 115卷 / 24期

关键词：

D O I：

10.1021/ja00077a047

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A concise total synthesis of (+)-piperazinomycin (1), a novel naturally occurring macrocyclic piperazine possessing antimicrobial and antifungal activity, is detailed with implementation of an improved Ullmann macrocyclization reaction conducted on a diketopiperazine (53%)

引用

页码：11426 / 11433

页数：8

共 58 条

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