THEORETICAL CONSIDERATIONS IN THE CALCULATION OF BIOAVAILABILITY OF DRUGS EXHIBITING MICHAELIS-MENTEN ELIMINATION KINETICS

被引:25
作者
RUBIN, GM [1 ]
TOZER, TN [1 ]
机构
[1] UNIV CALIF SAN FRANCISCO,DEPT PHARM,SAN FRANCISCO,CA 94143
来源
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS | 1984年 / 12卷 / 04期
关键词
D O I
10.1007/BF01062667
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:437 / 450
页数:14
相关论文
共 14 条
[1]   MODELS OF HEPATIC DRUG CLEARANCE - DISCRIMINATION BETWEEN THE WELL STIRRED AND PARALLEL-TUBE MODELS [J].
AHMAD, AB ;
BENNETT, PN ;
ROWLAND, M .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1983, 35 (04) :219-224
[2]   NONLINEAR ASSESSMENT OF PHENYTOIN BIOAVAILABILITY [J].
JUSKO, WJ ;
KOUP, JR ;
ALVAN, G .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1976, 4 (04) :327-336
[3]  
KEIDING S, 1978, J PHARMACOL EXP THER, V205, P465
[4]   1ST-PASS EFFECT - NON-LINEAR CONCEPT COMPRISING AN EXPLICIT SOLUTION OF INTEGRATED MICHAELIS-MENTEN EQUATION [J].
KELLER, F ;
SCHOLLE, J .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1981, 70 (02) :195-198
[5]   BIOAVAILABILITY CALCULATIONS FOR DRUGS SHOWING SIMULTANEOUS FIRST-ORDER AND CAPACITY-LIMITED ELIMINATION KINETICS [J].
MARTIS, L ;
LEVY, RH .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1973, 1 (04) :283-294
[6]  
MCLEAN AJ, 1978, CLIN PHARMACOL THER, V24, P5
[7]   EFFECT OF ALTERED PLASMA-PROTEIN BINDING ON APPARENT VOLUME OF DISTRIBUTION [J].
OIE, S ;
TOZER, TN .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1979, 68 (09) :1203-1205
[8]  
Pang K S, 1977, J Pharmacokinet Biopharm, V5, P625, DOI 10.1007/BF01059688
[9]  
Pang K S, 1977, J Pharmacokinet Biopharm, V5, P655, DOI 10.1007/BF01059689
[10]  
RIEGELMAN S, 1973, J PHARMACOKIN BIOPHA, V1, P418