PROBLEMS ASSOCIATED WITH THE APPLICATION OF THE CHENG-PRUSOFF RELATIONSHIP TO ESTIMATE ATROPINE AFFINITY CONSTANTS USING FUNCTIONAL TISSUE RESPONSES

被引:10
作者
EGLEN, RM
WHITING, RL
机构
关键词
D O I
10.1016/0024-3205(89)90221-X
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:81 / 94
页数:14
相关论文
共 21 条
[11]   COMPARISON OF DISSOCIATION CONSTANTS AND OF RELATIVE EFFICACIES OF SELECTED AGONISTS ACTING ON PARASYMPATHETIC RECEPTORS [J].
FURCHGOTT, RF ;
BURSZTYN, P .
ANNALS OF THE NEW YORK ACADEMY OF SCIENCES, 1967, 144 (A2) :882-+
[12]  
FURCHGOTT RF, 1984, TRENDS PHARM SCI S, V5, P45
[13]  
GIL DW, 1985, J PHARMACOL EXP THER, V232, P608
[14]  
KENAKIN TP, 1984, PHARMACOL REV, V36, P165
[15]   FUNCTIONAL AND DIRECT BINDING-STUDIES USING SUBTYPE SELECTIVE MUSCARINIC RECEPTOR ANTAGONISTS [J].
KUNYSZ, EL ;
MICHEL, AD ;
WHITING, RL .
BRITISH JOURNAL OF PHARMACOLOGY, 1988, 93 (03) :491-500
[16]  
LAZARENO S, 1986, IN PRESS P INT S MUS
[17]  
PENNEFATHER P, 1982, MOL PHARMACOL, V22, P369
[18]   KINETICS OF ACTION OF ACETYLCHOLINE ANTAGONISTS IN SMOOTH MUSCLE [J].
RANG, HP .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1966, 164 (996) :488-+
[19]   IMPORTANT CONCEPTS OF RECEPTOR THEORY [J].
RUFFOLO, RR .
JOURNAL OF AUTONOMIC PHARMACOLOGY, 1982, 2 (04) :277-295