CHIRAL N-PROTECTED BETA-IODOAMINES FROM ALPHA-AMINO-ACIDS - A GENERAL-SYNTHESIS

被引：31

作者：

CAPUTO, R ^{[1
]}

CASSANO, E ^{[1
]}

LONGOBARDO, L ^{[1
]}

PALUMBO, G ^{[1
]}

机构：

[1] UNIV NAPLES FEDERICO II,DIPARTIMENTO CHIM ORGAN & BIOL,I-80134 NAPLES,ITALY

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 01期

关键词：

D O I：

10.1016/0040-4039(94)02202-M

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

N-Protected D- or L-beta-iodoamines (as 2), which are useful intermediates for the preparation of chiral beta-aminoacids, are obtained smoothly from beta-aminols (as 1) in two steps and high yields.

引用

页码：167 / 168

页数：2

共 9 条

[1]

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[2]

CAPUTO R, 1994, IN PRESS SYNTHESIS

[3]

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[4]

ELMARINI A, 1992, SYNTHESIS-STUTTGART, P1104

[5]

Juaristi E., 1994, ALDRICHIM ACTA, V27, P3

[6]

KOKOTOS G, 1990, SYNTHESIS-STUTTGART, P299

[7]

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[8] A FACILE SYNTHESIS OF CHIRAL N-PROTECTED BETA-AMINO ALCOHOLS [J].

RODRIGUEZ, M ;

LLINARES, M ;

DOULUT, S ;

HEITZ, A ;

MARTINEZ, J .

TETRAHEDRON LETTERS, 1991, 32 (07) :923-926

[9] THE SYNTHESIS OF EITHER (+) OR (-) TRANS-2,5-DIMETHYLPYRROLIDINE [J].

SCHLESSINGER, RH ;

IWANOWICZ, EJ .

TETRAHEDRON LETTERS, 1987, 28 (19) :2083-2086

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