THE EFFECT OF TEMPERATURE ON CL-218872 AND PROPYL BETA-CARBOLINE-3-CARBOXYLATE INHIBITION OF [H-3]-LABELED FLUNITRAZEPAM BINDING IN RAT-BRAIN

被引:21
作者
GEE, KW
MORELLI, M
YAMAMURA, HI
机构
[1] UNIV ARIZONA, ARIZONA HLTH SCI CTR, DEPT BIOCHEM, TUCSON, AZ 85724 USA
[2] UNIV ARIZONA, ARIZONA HLTH SCI CTR, DEPT PSYCHIAT, TUCSON, AZ 85724 USA
[3] UNIV ARIZONA, ARIZONA HLTH SCI CTR, ARIZONA RES LABS, TUCSON, AZ 85724 USA
关键词
D O I
10.1016/0006-291X(82)90962-7
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1532 / 1537
页数:6
相关论文
共 14 条
[1]  
CHIU TH, 1982, MOL PHARMACOL, V21, P57
[2]  
EHLERT FJ, 1981, LIFE SCI, V29, P235, DOI 10.1016/0024-3205(81)90239-3
[3]  
EHLERT FJ, 1982, ADV PSYCHOPHARMACOLO
[4]   RESOLUTION OF 2 BIOCHEMICALLY AND PHARMACOLOGICALLY DISTINCT BENZODIAZEPINE RECEPTORS [J].
KLEPNER, CA ;
LIPPA, AS ;
BENSON, DI ;
SANO, MC ;
BEER, B .
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1979, 11 (04) :457-462
[5]   BENZODIAZEPINE RECEPTORS - CELLULAR AND BEHAVIORAL-CHARACTERISTICS [J].
LIPPA, AS ;
CRITCHETT, D ;
SANO, MC ;
KLEPNER, CA ;
GREENBLATT, EN ;
COUPET, J ;
BEER, B .
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1979, 10 (05) :831-843
[6]   PHYSICAL SEPARATION AND CHARACTERIZATION OF 2 TYPES OF BENZODIAZEPINE RECEPTORS [J].
LO, MMS ;
STRITTMATTER, SM ;
SNYDER, SH .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1982, 79 (02) :680-684
[7]   AGONIST AND ANTAGONIST BENZODIAZEPINE RECEPTOR INTERACTION INVITRO [J].
MOHLER, H ;
RICHARDS, JG .
NATURE, 1981, 294 (5843) :763-765
[8]   [PROPYL-H-3 BETA-CARBOLINE-3-CARBOXYLATE BINDS SPECIFICALLY TO BRAIN BENZODIAZEPINE RECEPTORS [J].
NIELSEN, M ;
SCHOU, H ;
BRAESTRUP, C .
JOURNAL OF NEUROCHEMISTRY, 1981, 36 (01) :276-285
[9]   BENZODIAZEPINE BINDING IN HUMAN-BRAIN - CHARACTERIZATION USING [H-3]FLUNITRAZEPAM [J].
SPETH, RC ;
WASTEK, GJ ;
JOHNSON, PC ;
YAMAMURA, HI .
LIFE SCIENCES, 1978, 22 (10) :859-866
[10]   BENZODIAZEPINE RECEPTORS - TEMPERATURE-DEPENDENCE OF [H-3] FLUNITRAZEPAM BINDING [J].
SPETH, RC ;
WASTEK, GJ ;
YAMAMURA, HI .
LIFE SCIENCES, 1979, 24 (04) :351-357