N-BENZYLTRIFLAMIDE - A GENERALLY USEFUL MITSUNOBU REAGENT FOR AMINE SYNTHESIS

被引：23

作者：

BELL, KE

KNIGHT, DW

GRAVESTOCK, MB

机构：

[1] UNIV NOTTINGHAM,DEPT CHEM,NOTTINGHAM NG7 2RD,ENGLAND

[2] ZENECA PHARMACEUT,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 47期

关键词：

D O I：

10.1016/0040-4039(95)01792-G

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

N-Benzyl triflamide has been found to be generally useful as a Mitsunobu nucleophile for the preparation of a range of primary and secondary benzylamines from the corresponding alcohols, using the standard reagents DEAD and triphenylphosphine.

引用

页码：8681 / 8684

页数：4

共 20 条

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