PEPTIDES DERIVED FROM KAINIC ACID AS ANTAGONISTS OF N-METHYL-D-ASPARTATE-INDUCED NEUROEXCITATION IN RAT-BRAIN

被引:8
作者
GOLDBERG, O [1 ]
TEICHBERG, VI [1 ]
机构
[1] WEIZMANN INST SCI,DEPT NEUROBIOL,IL-76100 REHOVOT,ISRAEL
关键词
D O I
10.1016/0304-3940(85)90388-X
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:101 / 105
页数:5
相关论文
共 23 条
[1]   D-ALPHA-AMINOADIPATE AS A SELECTIVE ANTAGONIST OF AMINO ACID-INDUCED AND SYNAPTIC EXCITATION OF MAMMALIAN SPINAL NEURONS [J].
BISCOE, TJ ;
EVANS, RH ;
FRANCIS, AA ;
MARTIN, MR ;
WATKINS, JC .
NATURE, 1977, 270 (5639) :743-745
[2]   EVALUATION OF D-ALPHA-AMINOADIPATE AND D-(AND DL-)ALPHA-AMINOSUBERATE AS SELECTIVE ANTAGONISTS OF EXCITATORY AMINO-ACIDS IN THE SUBSTANTIA NIGRA AND MESENCEPHALIC RETICULAR-FORMATION OF THE RAT [J].
COLLINGRIDGE, GL ;
DAVIES, J .
NEUROPHARMACOLOGY, 1979, 18 (02) :193-199
[3]   KAINIC ACID-DERIVATIVES WITH ANTICONVULSANT ACTIVITY [J].
COLLINS, JF ;
DIXON, AJ ;
BADMAN, G ;
DESARRO, G ;
CHAPMAN, AG ;
HART, GP ;
MELDRUM, BS .
NEUROSCIENCE LETTERS, 1984, 51 (03) :371-376
[4]   ANTICONVULSANT ACTION OF EXCITATORY AMINO-ACID ANTAGONISTS [J].
CROUCHER, MJ ;
COLLINS, JF ;
MELDRUM, BS .
SCIENCE, 1982, 216 (4548) :899-901
[5]   DIFFERENTIAL ACTIVATION AND BLOCKADE OF EXCITATORY AMINO-ACID RECEPTORS IN THE MAMMALIAN AND AMPHIBIAN CENTRAL NERVOUS SYSTEMS [J].
DAVIES, J ;
EVANS, RH ;
JONES, AW ;
SMITH, DAS ;
WATKINS, JC .
COMPARATIVE BIOCHEMISTRY AND PHYSIOLOGY C-PHARMACOLOGY TOXICOLOGY & ENDOCRINOLOGY, 1982, 72 (02) :211-224
[6]   2-AMINO-5-PHOSPHONOVALERATE(2APV), A POTENT AND SELECTIVE ANTAGONIST OF AMINO ACID-INDUCED AND SYNAPTIC EXCITATION [J].
DAVIES, J ;
FRANCIS, AA ;
JONES, AW ;
WATKINS, JC .
NEUROSCIENCE LETTERS, 1981, 21 (01) :77-81
[7]   ANTICONVULSANT PROPERTIES OF 3-HYDROXY-2-QUINOXALINECARBOXYLIC ACID, A NEWLY FOUND ANTAGONIST OF EXCITATORY AMINO-ACIDS [J].
EREZ, U ;
FRENK, H ;
GOLDBERG, O ;
COHEN, A ;
TEICHBERG, VI .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 110 (01) :31-39
[8]   ANTAGONISM OF EXCITATORY AMINO ACID-INDUCED RESPONSES AND OF SYNAPTIC EXCITATION IN THE ISOLATED SPINAL-CORD OF THE FROG [J].
EVANS, RH ;
FRANCIS, AA ;
HUNT, K ;
OAKES, DJ ;
WATKINS, JC .
BRITISH JOURNAL OF PHARMACOLOGY, 1979, 67 (04) :591-603
[9]   THE EFFECTS OF A SERIES OF OMEGA-PHOSPHONIC ALPHA-CARBOXYLIC AMINO-ACIDS ON ELECTRICALLY EVOKED AND EXCITANT AMINO ACID-INDUCED RESPONSES IN ISOLATED SPINAL-CORD PREPARATIONS [J].
EVANS, RH ;
FRANCIS, AA ;
JONES, AW ;
SMITH, DAS ;
WATKINS, JC .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 75 (01) :65-75
[10]   DIPEPTIDE ANTAGONISTS OF AMINO ACID-INDUCED AND SYNAPTIC EXCITATION IN THE FROG SPINAL-CORD [J].
FRANCIS, AA ;
JONES, AW ;
WATKINS, JC .
JOURNAL OF NEUROCHEMISTRY, 1980, 35 (06) :1458-1460