DETERMINATION OF BIOLOGICAL-ACTIVITY OF ADINAZOLAM AND ITS METABOLITES

被引:32
作者
SETHY, VH
COLLINS, RJ
DANIELS, EG
机构
关键词
D O I
10.1111/j.2042-7158.1984.tb04449.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
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页码:546 / 548
页数:3
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共 11 条
[1]   PARTIAL AGONISTS FOR BRAIN GABA-BENZODIAZEPINE RECEPTOR COMPLEX [J].
BRAESTRUP, C ;
NIELSEN, M ;
KROGSGAARDLARSEN, P ;
FALCH, E .
NATURE, 1979, 280 (5720) :331-333
[2]   GABA REDUCES BINDING OF H-3-LABELED METHYL BETA-CARBOLINE-3-CARBOXYLATE TO BRAIN BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M .
NATURE, 1981, 294 (5840) :472-474
[3]  
Braestrup C., 1982, PHARM BENZODIAZEPINE, P71
[4]   PHARMACOLOGY OF SOME METABOLITES OF TRIAZOLAM, ALPRAZOLAM, AND DIAZEPAM PREPARED BY A SIMPLE, ONE-STEP OXIDATION OF BENZODIAZEPINES [J].
GALL, M ;
KAMDAR, BV ;
COLLINS, RJ .
JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (12) :1290-1294
[5]   1-(AMINOALKYL)-6-ARYL-4H-S-TRIAZOLO[4,3-A][1,4]BENZODIAZEPINES WITH ANTIANXIETY AND ANTI-DEPRESSANT ACTIVITY [J].
HESTER, JB ;
RUDZIK, AD ;
VONVOIGTLANDER, PF .
JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (04) :392-402
[6]  
LAHTI RA, 1982, SOC NEUR ABSTS, V8, P463
[7]  
MOFFETT RB, 1978, J MED CHEM, V21, P1290
[8]  
PYKE RE, 1983, PSYCHOPHARMACOL BULL, V19, P96
[9]   INTERACTION OF TRIAZOLOBENZODIAZEPINES WITH BENZODIAZEPINE RECEPTORS [J].
SETHY, VH ;
RUSSELL, RR ;
DAENZER, CL .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1983, 35 (08) :524-526
[10]   DETERMINATION OF BIOLOGICAL-ACTIVITY OF ALPRAZOLAM, TRIAZOLAM AND THEIR METABOLITES [J].
SETHY, VH ;
HARRIS, DW .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1982, 34 (02) :115-116