THE ROLE OF THE BENZODIAZEPINE RECEPTOR IN MEDIATING LONG-LASTING ANTICONVULSANT EFFECTS AND THE LATE-APPEARING REDUCTIONS IN MOTOR-ACTIVITY AND EXPLORATION

被引:5
作者
FILE, SE [1 ]
WILKS, LJ [1 ]
MABBUTT, PS [1 ]
机构
[1] UNIV LONDON, SCH PHARM, MRC, NEUROPHARMACOL RES GRP, LONDON WC1N 1AX, ENGLAND
基金
英国惠康基金;
关键词
D O I
10.1007/BF00439449
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:349 / 354
页数:6
相关论文
共 15 条
[1]   BENZODIAZEPINE ANTAGONIST RO 15-1788 - NEUROLOGICAL AND BEHAVIORAL-EFFECTS [J].
BONETTI, EP ;
PIERI, L ;
CUMIN, R ;
SCHAFFNER, R ;
PIERI, M ;
GAMZU, ER ;
MULLER, RKM ;
HAEFELY, W .
PSYCHOPHARMACOLOGY, 1982, 78 (01) :8-18
[2]   PHARMACOKINETIC MODELING OF THE ANTICONVULSANT RESPONSE OF OXAZEPAM IN RATS USING THE PENTYLENETETRAZOL THRESHOLD CONCENTRATION AS PHARMACODYNAMIC MEASURE [J].
DINGEMANSE, J ;
SOLLIE, FAE ;
BREIMER, DD ;
DANHOF, M .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1988, 16 (02) :203-228
[4]   LONG-LASTING ANTICONVULSANT EFFECTS OF DIAZEPAM IN DIFFERENT MOUSE STRAINS - CORRELATIONS WITH BRAIN CONCENTRATIONS AND RECEPTOR OCCUPANCY [J].
FILE, SE ;
GREENBLATT, DJ ;
MARTIN, IL ;
BROWN, C .
PSYCHOPHARMACOLOGY, 1985, 86 (1-2) :137-141
[5]   RELIABILITY OF HOLE-BOARD APPARATUS [J].
FILE, SE ;
WARDILL, AG .
PSYCHOPHARMACOLOGIA, 1975, 44 (01) :47-51
[6]   BEHAVIORAL PHARMACOLOGY OF MINOR TRANQUILIZERS [J].
FILE, SE ;
PELLOW, S .
PHARMACOLOGY & THERAPEUTICS, 1987, 35 (03) :265-290
[7]  
HAEFELY WE, 1987, CHIMIA, V41, P389
[8]   SELECTIVE ANTAGONISTS OF BENZODIAZEPINES [J].
HUNKELER, W ;
MOHLER, H ;
PIERI, L ;
POLC, P ;
BONETTI, EP ;
CUMIN, R ;
SCHAFFNER, R ;
HAEFELY, W .
NATURE, 1981, 290 (5806) :514-516
[9]   METHODS FOR THE DETERMINATION OF LORAZEPAM AND CHLORDIAZEPOXIDE AND METABOLITES IN BRAIN-TISSUE - A COMPARISON WITH PLASMA-CONCENTRATIONS IN THE RAT [J].
LISTER, RG ;
ABERNETHY, DR ;
GREENBLATT, DJ ;
FILE, SE .
JOURNAL OF CHROMATOGRAPHY, 1983, 277 (OCT) :201-208
[10]  
LISTER RG, 1987, PSYCHOPHARMACOLOGY, V92, P180