2-AZA-1,3-DIENES - A NEW AND SIMPLE METHOD FOR THE SYNTHESIS OF FUNCTIONALIZED PYRIDINE-DERIVATIVES

被引：17

作者：

BARLUENGA, J ^{[1
]}

GONZALEZ, FJ ^{[1
]}

CARLON, RP ^{[1
]}

FUSTERO, S ^{[1
]}

机构：

[1] UNIV VALENCIA, FAC FARM, DEPT QUIM ORGAN, E-46010 VALENCIA, SPAIN

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1991年 / 56卷 / 24期

关键词：

D O I：

10.1021/jo00024a011

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of 4(1H)-pyridones and 4-chloropyridines from 2-aza 1,3-dienes is described, using carbonic acid derivatives. The process involves a [5 + 1] heterocyclization reaction, with formation of two new carbon-carbon bonds.

引用

页码：6751 / 6754

页数：4

共 35 条

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[2] REACTIONS OF KETIMINES AND ETHYL PHENYLPROPIOLATE - SYNTHESIS OF 4-OXODIHYDROPYRIDINES
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[4] AN EFFICIENT AND GENERAL STRATEGY FOR THE SYNTHESIS OF 1,4-DIHYDRO-LAMBDA-3-AZAPHOSPHININES AND 1,4-DIHYDRO-LAMBDA-5-AZAPHOSPHININES FROM 2-AZA-1,3-DIENES
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[5] DIELS-ALDER REACTION OF UNACTIVATED 2-AZA-1,3-DIENES WITH DIETHYL KETOMALONATE - A CARBON-DIOXIDE EQUIVALENT
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FUSTERO, S
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[6] SYNTHESIS OF 4(1H)-PYRIDONES BY CARBONYLATION OF 2-AZA-1,3-DIENES
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[8] PREPARATION AND REACTIVITY OF 2-AZA-1,3-BUTADIENES - A DIELS-ALDER ROUTE TO 5,6-DIHYDRO-2H-1,3-OXAZINE DERIVATIVES
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[9] NEW PERSPECTIVES OF CARBO-1,3-DIENES AND HETERO-1,3-DIENES IN ORGANIC-SYNTHESIS
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