A VERY HIGH-AFFINITY OPIOID BINDING-SITE IN RAT-BRAIN - DEMONSTRATION BY COMPUTER MODELING

被引:64
作者
LUTZ, RA
CRUCIANI, RA
COSTA, T
MUNSON, PJ
RODBARD, D
机构
关键词
D O I
10.1016/0006-291X(84)90469-8
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
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页码:265 / 269
页数:5
相关论文
共 10 条
[1]   NALOXAZONE IRREVERSIBLY INHIBITS THE HIGH-AFFINITY BINDING OF [I-125]D-ALA2-D-LEU5-ENKEPHALIN [J].
HAZUM, E ;
CHANG, KJ ;
CUATRECASAS, P ;
PASTERNAK, GW .
LIFE SCIENCES, 1981, 28 (26) :2973-2979
[2]   LIGAND - A VERSATILE COMPUTERIZED APPROACH FOR CHARACTERIZATION OF LIGAND-BINDING SYSTEMS [J].
MUNSON, PJ ;
RODBARD, D .
ANALYTICAL BIOCHEMISTRY, 1980, 107 (01) :220-239
[3]  
NISHIMURA SL, 1984, MOL PHARMACOL, V25, P29
[4]   OPIATE ANALGESIA - EVIDENCE FOR MEDIATION BY A SUB-POPULATION OF OPIATE RECEPTORS [J].
PASTERNAK, GW ;
CHILDERS, SR ;
SNYDER, SH .
SCIENCE, 1980, 208 (4443) :514-516
[5]   IDENTIFICATION OF NOVEL HIGH AFFINITY OPIATE RECEPTOR-BINDING IN RAT-BRAIN [J].
PASTERNAK, GW ;
SNYDER, SH .
NATURE, 1975, 253 (5492) :563-565
[6]  
PASTERNAK GW, 1980, J PHARMACOL EXP THER, V214, P455
[7]  
PASTERNAK GW, 1980, J MED CHEM, V23, P674, DOI 10.1021/jm00180a019
[8]   PROLACTIN AND GROWTH-HORMONE RELEASE BY MORPHINE IN THE RAT - DIFFERENT RECEPTOR MECHANISMS [J].
SPIEGEL, K ;
KOURIDES, IA ;
PASTERNAK, GW .
SCIENCE, 1982, 217 (4561) :745-747
[9]  
ZHANG AZ, 1981, LIFE SCI, V29, P843
[10]   ONTOGENY OF OPIOID PHARMACOLOGY AND RECEPTORS - HIGH AND LOW AFFINITY SITE DIFFERENCES [J].
ZHANG, AZ ;
PASTERNAK, GW .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 73 (01) :29-40