Structure and pharmacology of vertebrate GABA(A) receptor subtypes

被引:183
作者
Whiting, PJ
Mckernan, RM
Wafford, KA
机构
[1] Neuroscience Research Centre, Merck Sharp & Dohme, Harlow
来源
INTERNATIONAL REVIEW OF NEUROBIOLOGY, VOL 38 | 1995年 / 38卷
关键词
D O I
10.1016/S0074-7742(08)60525-5
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:95 / 138
页数:44
相关论文
共 209 条
[81]   THE GAMMA-3-SUBUNIT OF THE GABA-A-RECEPTOR CONFERS SENSITIVITY TO BENZODIAZEPINE RECEPTOR LIGANDS [J].
KNOFLACH, F ;
RHYNER, T ;
VILLA, M ;
KELLENBERGER, S ;
DRESCHER, U ;
MALHERBE, P ;
SIGEL, E ;
MOHLER, H .
FEBS LETTERS, 1991, 293 (1-2) :191-194
[82]   PHARMACOLOGICAL AND ELECTROPHYSIOLOGICAL PROPERTIES OF RECOMBINANT GABA-A-RECEPTORS COMPRISING THE ALPHA-3-SUBUNIT, BETA-1-SUBUNIT AND GAMMA-2-SUBUNIT [J].
KNOFLACH, F ;
BACKUS, KH ;
GILLER, T ;
MALHERBE, P ;
PFLIMLIN, P ;
MOHLER, H ;
TRUBE, G .
EUROPEAN JOURNAL OF NEUROSCIENCE, 1992, 4 (01) :1-9
[83]   FISH ORDERING OF REFERENCE MARKERS AND OF THE GENE FOR THE ALPHA-5 SUBUNIT OF THE GAMMA-AMINOBUTYRIC-ACID RECEPTOR (GABRA5) WITHIN THE ANGELMAN AND PRADER-WILLI SYNDROME CHROMOSOMAL REGIONS [J].
KNOLL, JHM ;
SINNETT, D ;
WAGSTAFF, J ;
GLATT, K ;
WILCOX, AS ;
WHITING, PM ;
WINGROVE, P ;
SIKELA, JM ;
LALANDE, M .
HUMAN MOLECULAR GENETICS, 1993, 2 (02) :183-189
[84]   GENERATION OF 2 FORMS OF THE GAMMA-AMINOBUTYRIC ACIDA RECEPTOR GAMMA-2-SUBUNIT IN MICE BY ALTERNATIVE SPLICING [J].
KOFUJI, P ;
JIA, BW ;
MOSS, SJ ;
HUGANIR, RL ;
BURT, DR .
JOURNAL OF NEUROCHEMISTRY, 1991, 56 (02) :713-715
[85]  
KORPI ER, 1993, MOL PHARMACOL, V44, P87
[86]  
KORPI ER, 1994, J NEUROCHEM, V63, P1167
[87]   REGULATION OF GABA(A) RECEPTOR FUNCTION BY PROTEIN-KINASE-C PHOSPHORYLATION [J].
KRISHEK, BJ ;
XIE, XM ;
BLACKSTONE, C ;
HUGANIR, RL ;
MOSS, SJ ;
SMART, TG .
NEURON, 1994, 12 (05) :1081-1095
[88]   EFFECT OF IVERMECTIN ON GAMMA-AMINOBUTYRIC ACID-INDUCED CHLORIDE CURRENTS IN MOUSE HIPPOCAMPAL EMBRYONIC NEURONS [J].
KRUSEK, J ;
ZEMKOVA, H .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1994, 259 (02) :121-128
[89]   GABA RHO-2 RECEPTOR PHARMACOLOGICAL PROFILE - GABA RECOGNITION SITE SIMILARITIES TO RHO-1 [J].
KUSAMA, T ;
WANG, TL ;
GUGGINO, WB ;
CUTTING, GR ;
UHL, GR .
EUROPEAN JOURNAL OF PHARMACOLOGY-MOLECULAR PHARMACOLOGY SECTION, 1993, 245 (01) :83-84
[90]   PHARMACOLOGY OF GABA RHO-1 AND GABA ALPHA/BETA RECEPTORS EXPRESSED IN XENOPUS OOCYTES AND COS CELLS [J].
KUSAMA, T ;
SPIVAK, CE ;
WHITING, P ;
DAWSON, VL ;
SCHAEFFER, JC ;
UHL, GR .
BRITISH JOURNAL OF PHARMACOLOGY, 1993, 109 (01) :200-206