DRUG-RECEPTOR INTERACTIONS - EXAMPLE OF CARDIAC GLYCOSIDE RECEPTORS OF ERYTHROCYTE-MEMBRANE

被引:2
作者
ERDMANN, E [1 ]
机构
[1] UNIV MUNICH, KLINIKUM GROSSHADERN, MED KLIN 1, MARCHIONINISTRASSE 15, 8000 MUNICH, GERMANY
来源
BLUT | 1976年 / 32卷 / 02期
关键词
D O I
10.1007/BF00995933
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
This is a review of the molecular kinetics on the inhibition of active Na transport by cardiac glycosides, the equilibrium of the ouabain-receptor complex, cardiac glycoside receptor binding in human erythrocyte membrane and the receptor density per erythrocyte.
引用
收藏
页码:61 / 70
页数:10
相关论文
共 62 条
[41]   EFFECTS OF N-ACETYLIMIDAZOLE ON HUMAN ERYTHROCYTE ATPASE ACTIVITY - EVIDENCE FOR A TYROSYL RESIDUE AT ATP BINDING-SITE OF (NA++K+)-DEPENDENT ATPASE [J].
MASIAK, SJ ;
DANGELO, G .
BIOCHIMICA ET BIOPHYSICA ACTA, 1975, 382 (01) :83-91
[42]   MECHANISM OF CARDIAC GLYCOSIDE INHIBITION OF (NA+-K+)-DEPENDENT ATPASE FROM CARDIAC TISSUE [J].
MATSUI, H ;
SCHWARTZ, A .
BIOCHIMICA ET BIOPHYSICA ACTA, 1968, 151 (03) :655-&
[43]  
MIRCEVOVA L, 1973, Folia Haematologica (Leipzig), V99, P317
[44]  
MOORE WV, 1974, J BIOL CHEM, V249, P6255
[45]  
MUELLER TJ, 1974, J BIOL CHEM, V249, P7568
[46]   PATHOLOGICAL ALTERATIONS OF CATION MOVEMENTS IN RED BLOOD-CELLS [J].
PARKER, JC ;
WELT, LG .
ARCHIVES OF INTERNAL MEDICINE, 1972, 129 (02) :320-+
[47]  
PATSERNAK GW, 1974, MOL PHARMACOL, V10, P183
[48]   RESOLUTION OF PUMP AND LEAK COMPONENTS OF SODIUM AND POTASSIUM ION TRANSPORT IN HUMAN ERYTHROCYTES [J].
POST, RL ;
ALBRIGHT, CD ;
DAYANI, K .
JOURNAL OF GENERAL PHYSIOLOGY, 1967, 50 (05) :1201-+
[49]   INTERACTION OF EXTERNAL K, NA, AND CARDIOACTIVE STEROIDS WITH NA-K PUMP OF HUMAN RED BLOOD-CELL [J].
SACHS, JR .
JOURNAL OF GENERAL PHYSIOLOGY, 1974, 63 (02) :123-143
[50]   THE ATTRACTIONS OF PROTEINS FOR SMALL MOLECULES AND IONS [J].
SCATCHARD, G .
ANNALS OF THE NEW YORK ACADEMY OF SCIENCES, 1949, 51 (04) :660-672