CONFORMATIONALLY CONSTRAINED NONPEPTIDE BETA-TURN MIMETICS OF ENKEPHALIN

被引：102

作者：

GARDNER, B

NAKANISHI, H

KAHN, M

机构：

[1] MOLECUMET INST,2023 120TH AVE NE,BELLEVUE,WA 98005

[2] UNIV WASHINGTON,DEPT PATHOBIOL,SEATTLE,WA 98195

[3] UNIV ILLINOIS,DEPT CHEM,CHICAGO,IL 60680

来源：

TETRAHEDRON | 1993年 / 49卷 / 17期

关键词：

D O I：

10.1016/S0040-4020(01)90205-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The design synthesis and in vitro biological analysis of a family of conformationally constrained nonpeptide mimetics incorporating a 4-->1 beta-turn prosthetic unit to examine the proposed biological significance of this conformer is described.

引用

页码：3433 / 3448

页数：16

共 40 条

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