BENZODIAZEPINE AGONIST-TYPE ACTIVITY OF RAUBASINE, A RAUWOLFIA SERPENTINA ALKALOID

被引:8
作者
CHARVERON, M [1 ]
ASSIE, MB [1 ]
STENGER, A [1 ]
BRILEY, M [1 ]
机构
[1] CTR RECH PIERRE FABRE,DEPT BIOCHEM PHARMACOL,17 AVE JEAN MOULIN,F-81106 CASTRES,FRANCE
关键词
D O I
10.1016/0014-2999(84)90718-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:313 / 317
页数:5
相关论文
共 18 条
[1]   INVITRO AND INVIVO INHIBITION BY ZOPICLONE OF BENZODIAZEPINE BINDING TO RODENT BRAIN RECEPTORS [J].
BLANCHARD, JC ;
BOIREAU, A ;
GARRET, C ;
JULOU, L .
LIFE SCIENCES, 1979, 24 (26) :2417-2420
[2]   SURICLONE - A NEW CYCLOPYRROLONE DERIVATIVE RECOGNIZING RECEPTORS LABELED BY BENZODIAZEPINES IN RAT HIPPOCAMPUS AND CEREBELLUM [J].
BLANCHARD, JC ;
JULOU, L .
JOURNAL OF NEUROCHEMISTRY, 1983, 40 (03) :601-607
[3]   INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SCHMIECHEN, R ;
NEEF, G ;
NIELSEN, M ;
PETERSEN, EN .
SCIENCE, 1982, 216 (4551) :1241-1243
[4]  
CARMINES EL, 1980, J ENVIRON PATHOL TOX, V4, P23
[5]  
CARVALHO LP, 1983, NATURE, V301, P64
[6]   BENZODIAZEPINE RECEPTORS - LABELING IN INTACT ANIMALS WITH [H-3]FLUNITRAZEPAM [J].
CHANG, RSL ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 48 (02) :213-218
[7]   CGS-8216 - RECEPTOR-BINDING CHARACTERISTICS OF A POTENT BENZODIAZEPINE ANTAGONIST [J].
CZERNIK, AJ ;
PETRACK, B ;
KALINSKY, HJ ;
PSYCHOYOS, S ;
CASH, WD ;
TSAI, C ;
RINEHART, RK ;
GRANAT, FR ;
LOVELL, RA ;
BRUNDISH, DE ;
WADE, R .
LIFE SCIENCES, 1982, 30 (04) :363-372
[8]   A NOVEL PYRAZOLOQUINOLINE THAT INTERACTS WITH BRAIN BENZODIAZEPINE RECEPTORS - CHARACTERIZATION OF SOME INVITRO AND INVIVO PROPERTIES OF CGS-9896 [J].
GEE, KW ;
YAMAMURA, HI .
LIFE SCIENCES, 1982, 30 (26) :2245-2252
[9]   CONVULSIONS INDUCED BY SUBMAXIMAL DOSE OF PENTYLENETETRAZOL IN MICE ARE ANTAGONIZED BY THE BENZODIAZEPINE ANTAGONIST RO 15-1788 [J].
GRECKSCH, G ;
DECARVALHO, LP ;
VENAULT, P ;
CHAPOUTHIER, G ;
ROSSIER, J .
LIFE SCIENCES, 1983, 32 (22) :2579-2584
[10]   SELECTIVE ANTAGONISTS OF BENZODIAZEPINES [J].
HUNKELER, W ;
MOHLER, H ;
PIERI, L ;
POLC, P ;
BONETTI, EP ;
CUMIN, R ;
SCHAFFNER, R ;
HAEFELY, W .
NATURE, 1981, 290 (5806) :514-516