PRACTICAL EPC SYNTHESIS OF 1,2-AMINO AND 1,3-AMINO ALCOHOLS

被引：19

作者：

GMEINER, P

KARTNER, A

JUNGE, D

机构：

[1] Institut für Pharmazie, Lebensmittelchemie der Ludwig-Maximilians-Universität, D-8000 München 2

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 27期

关键词：

D O I：

10.1016/S0040-4039(00)79340-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient synthesis of enantiomerically pure 1,2- and 1,3-amino alcohols (4, 10) through the key intermediates 2 and 8a,b, obtained from L-aspartic acid, is reported. Using 4d as an example it is shown that the products can serve as precursors for unusual amino aldehydes and nonproteinogenic amino acids.

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页码：4325 / 4326

页数：2

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