INVIVO DETERMINATION OF THE PROFILE OF BENZODIAZEPINE LIGANDS BY COMPARING THE INHIBITION OF H-3 RO-15-1788 BINDING TO THE MODULATION OF CGMP LEVELS IN MOUSE CEREBELLUM

被引:6
作者
BOIREAU, A
MARTEL, M
FARGES, G
DUBEDAT, P
LADURON, PM
BLANCHARD, JC
机构
关键词
D O I
10.1016/0006-2952(88)90413-3
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:3765 / 3769
页数:5
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共 32 条
  • [1] PHARMACOLOGICAL PROFILE OF THE IMIDAZOPYRIDINE ZOLPIDEM AT BENZODIAZEPINE RECEPTORS AND ELECTROCORTICOGRAM IN RATS
    ARBILLA, S
    DEPOORTERE, H
    GEORGE, P
    LANGER, SZ
    [J]. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1985, 330 (03) : 248 - 251
  • [2] SUPPRESSION OF INHIBITION IN CEREBELLAR CORTEX BY PICROTOXIN AND BICUCULLINE
    BISTI, S
    IOSIF, G
    STRATA, P
    [J]. BRAIN RESEARCH, 1971, 28 (03) : 591 - &
  • [3] INVITRO AND INVIVO INHIBITION BY ZOPICLONE OF BENZODIAZEPINE BINDING TO RODENT BRAIN RECEPTORS
    BLANCHARD, JC
    BOIREAU, A
    GARRET, C
    JULOU, L
    [J]. LIFE SCIENCES, 1979, 24 (26) : 2417 - 2420
  • [4] INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS
    BRAESTRUP, C
    SCHMIECHEN, R
    NEEF, G
    NIELSEN, M
    PETERSEN, EN
    [J]. SCIENCE, 1982, 216 (4551) : 1241 - 1243
  • [5] LIGANDS FOR BENZODIAZEPINE RECEPTORS WITH POSITIVE AND NEGATIVE EFFICACY
    BRAESTRUP, C
    HONORE, T
    NIELSEN, M
    PETERSEN, EN
    JENSEN, LH
    [J]. BIOCHEMICAL PHARMACOLOGY, 1984, 33 (06) : 859 - 862
  • [6] Braestrup C, 1986, BENZODIAZEPINE GABA, P167
  • [7] THE BENZODIAZEPINE ANTAGONIST RO-15-1788 REVERSES THE EFFECT OF "METHYL-BETA-CARBOLINE-3-CARBOXYLATE BUT NOT OF HARMALINE ON CEREBELLAR CGMP AND MOTOR-PERFORMANCE IN MICE
    BURKARD, WP
    BONETTI, EP
    HAEFELY, W
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 109 (02) : 241 - 247
  • [8] GABA, BICUCULLINE AND CENTRAL INHIBITION
    CURTIS, DR
    DUGGAN, AW
    FELIX, D
    JOHNSTON, GA
    [J]. NATURE, 1970, 226 (5252) : 1222 - &
  • [9] CGS-8216 - RECEPTOR-BINDING CHARACTERISTICS OF A POTENT BENZODIAZEPINE ANTAGONIST
    CZERNIK, AJ
    PETRACK, B
    KALINSKY, HJ
    PSYCHOYOS, S
    CASH, WD
    TSAI, C
    RINEHART, RK
    GRANAT, FR
    LOVELL, RA
    BRUNDISH, DE
    WADE, R
    [J]. LIFE SCIENCES, 1982, 30 (04) : 363 - 372
  • [10] A NOVEL PYRAZOLOQUINOLINE THAT INTERACTS WITH BRAIN BENZODIAZEPINE RECEPTORS - CHARACTERIZATION OF SOME INVITRO AND INVIVO PROPERTIES OF CGS-9896
    GEE, KW
    YAMAMURA, HI
    [J]. LIFE SCIENCES, 1982, 30 (26) : 2245 - 2252