CGS-9896 - A NONBENZODIAZEPINE, NONSEDATING POTENTIAL ANXIOLYTIC

被引：70

作者：

BENNETT, DA

PETRACK, B

机构：

来源：

DRUG DEVELOPMENT RESEARCH | 1984年 / 4卷 / 01期

关键词：

D O I：

10.1002/ddr.430040109

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：75 / 82

页数：8

共 31 条

[1]

[Anonymous], 1980, ANNU REP MED CHEM, DOI 10.1016/S0065-7743(08)60367-X

[2]

ATRENS DM, 1976, PSYCHOPHARMACOLOGY, V49, P97

[3]

BENNETT DA, 1983, PHARMACOLOGIST, V25, P155

[4]

BERNARD PS, 1983, FED PROC, V42, P345

[5] GABA REDUCES BINDING OF H-3-LABELED METHYL BETA-CARBOLINE-3-CARBOXYLATE TO BRAIN BENZODIAZEPINE RECEPTORS [J].

BRAESTRUP, C ;

NIELSEN, M .

NATURE, 1981, 294 (5840) :472-474

[6] SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION) [J].

BRAESTRUP, C ;

SQUIRES, RF .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) :3805-3809

[7]

Braestrup C, 1983, HDB PSYCHOPHARMACOLO, P285

[8] PHOTOAFFINITY-LABELING OF THE BENZODIAZEPINE RECEPTOR CANNOT BE USED TO PREDICT LIGAND EFFICACY [J].

BROWN, CL ;

MARTIN, IL .

NEUROSCIENCE LETTERS, 1983, 35 (01) :37-40

[9]

COOK L, 1973, BENZODIAZEPINES, P327

[10] HIGH-AFFINITY INHIBITION OF [H-3-LABELED FLUNITRAZEPAM BINDING TO BRAIN BENZODIAZEPINE RECEPTORS BY CGS 9896, A NOVEL PYRAZOLOQUINOLINE [J].

GEE, KW ;

HORST, WD ;

OBRIEN, R ;

YAMAMURA, HI .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 105 (02) :457-461

← 1 2 3 4 →