POTENTIATION BY THIORPHAN AND BESTATIN OF THE NALOXONE-INSENSITIVE ANALGESIC EFFECTS OF NEUROTENSIN AND NEUROMEDIN-N

被引:56
作者
COQUEREL, A [1 ]
DUBUC, I [1 ]
KITABGI, P [1 ]
COSTENTIN, J [1 ]
机构
[1] UNIV NICE, FAC SCI, CTR BIOCHIM, CNRS, F-06034 NICE, FRANCE
关键词
D O I
10.1016/0197-0186(88)90175-1
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:361 / 366
页数:6
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共 25 条
  • [1] HYPOTHERMIA AND INTOLERANCE TO COLD INDUCED BY INTRACISTERNAL ADMINISTRATION OF HYPOTHALAMIC PEPTIDE NEUROTENSIN
    BISSETTE, G
    NEMEROFF, CB
    LOOSEN, PT
    PRANGE, AJ
    LIPTON, MA
    [J]. NATURE, 1976, 262 (5569) : 607 - 609
  • [2] CARRAWAY R, 1973, J BIOL CHEM, V248, P6854
  • [3] THE USE OF RADIOIMMUNOASSAY TO COMPARE THE TISSUE AND SUBCELLULAR DISTRIBUTIONS OF NEUROTENSIN AND NEUROMEDIN-N IN THE CAT
    CARRAWAY, RE
    MITRA, SP
    [J]. ENDOCRINOLOGY, 1987, 120 (05) : 2092 - 2100
  • [4] DEGRADATION OF NEUROTENSIN BY RAT-BRAIN SYNAPTIC-MEMBRANES - INVOLVEMENT OF A THERMOLYSIN-LIKE METALLOENDOPEPTIDASE (ENKEPHALINASE), ANGIOTENSIN-CONVERTING ENZYME, AND OTHER UNIDENTIFIED PEPTIDASES
    CHECLER, F
    VINCENT, JP
    KITABGI, P
    [J]. JOURNAL OF NEUROCHEMISTRY, 1983, 41 (02) : 375 - 384
  • [5] NEUROMEDIN-N - HIGH-AFFINITY INTERACTION WITH BRAIN NEUROTENSIN RECEPTORS AND RAPID INACTIVATION BY BRAIN SYNAPTIC PEPTIDASES
    CHECLER, F
    VINCENT, JP
    KITABGI, P
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 126 (03) : 239 - 244
  • [6] INACTIVATION OF NEUROTENSIN BY RAT-BRAIN SYNAPTIC-MEMBRANES - CLEAVAGE AT THE PRO10-TYR11 BOND BY ENDOPEPTIDASE-24.11 (ENKEPHALINASE) AND A PEPTIDASE DIFFERENT FROM PROLINE-ENDOPEPTIDASE
    CHECLER, F
    EMSON, PC
    VINCENT, JP
    KITABGI, P
    [J]. JOURNAL OF NEUROCHEMISTRY, 1984, 43 (05) : 1295 - 1301
  • [7] NEUROTENSIN - ANTINOCISPONSIVE ACTION IN RODENTS
    CLINESCHMIDT, BV
    MCGUFFIN, JC
    BUNTING, PB
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 54 (1-2) : 129 - 139
  • [8] NALOXONE-INSENSITIVE POTENTIATION OF NEUROTENSIN HYPOTHERMIC EFFECT BY THE ENKEPHALINASE INHIBITOR THIORPHAN
    COQUEREL, A
    DUBUC, I
    MENARD, JF
    KITABGI, P
    COSTENTIN, J
    [J]. BRAIN RESEARCH, 1986, 398 (02) : 386 - 389
  • [9] DISSOCIATED EFFECTS OF INHIBITORS OF ENKEPHALIN-METABOLIZING PEPTIDASES OR NALOXONE ON VARIOUS NOCICEPTIVE RESPONSES
    COSTENTIN, J
    VLAICULESCU, A
    CHAILLET, P
    BENNATAN
    AVEAUX, D
    SCHWARTZ, JC
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 123 (01) : 37 - 44
  • [10] D'amour FE, 1941, J PHARMACOL EXP THER, V72, P74