INHIBITION OF PLATELET THROMBOXANE SYNTHESIS BY 7-(1-IMIDAZOLYL) HEPTANOIC ACID - DISSOCIATION FROM INHIBITION OF AGGREGATION

被引:56
作者
GRIMM, LJ
KNAPP, DR
SENATOR, D
HALUSHKA, PV
机构
[1] MED UNIV S CAROLINA,DEPT PHARMACOL,CHARLESTON,SC 29401
[2] MED UNIV S CAROLINA,DEPT MED,CHARLESTON,SC 29401
关键词
D O I
10.1016/0049-3848(81)90004-9
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:307 / 317
页数:11
相关论文
共 23 条
[1]   REGULATION OF POSTOCCLUSIVE HYPEREMIA BY ENDOGENOUSLY SYNTHESIZED PROSTAGLANDINS IN DOG HEART [J].
ALEXANDER, RW ;
KENT, KM ;
PISANO, JJ ;
KEISER, HR ;
COOPER, T .
JOURNAL OF CLINICAL INVESTIGATION, 1975, 55 (06) :1174-1181
[2]  
BERTELE, 1981, LANCET, V1, P1057
[3]  
BEST LC, 1980, THROMB HAEMOSTASIS, V43, P38
[4]   METABOLISM OF (C-14) ARACHIDONIC-ACID BY HUMAN PLATELETS [J].
BILLS, TK ;
SMITH, JB ;
SILVER, MJ .
BIOCHIMICA ET BIOPHYSICA ACTA, 1976, 424 (02) :303-314
[5]  
BLACKWELL GJ, 1978, BRIT J PHARMACOL, V64, pP435
[6]   AGGREGATION OF BLOOD PLATELETS BY ADENOSINE DIPHOSPHATE AND ITS REVERSAL [J].
BORN, GVR .
NATURE, 1962, 194 (4832) :927-&
[7]  
BURCH RM, 1979, J PHARMACOL EXP THER, V210, P344
[8]   VASOPRESSIN-STIMULATED WATER-FLOW IS DECREASED BY THROMBOXANE SYNTHESIS INHIBITION OR ANTAGONISM [J].
BURCH, RM ;
KNAPP, DR ;
HALUSHKA, PV .
AMERICAN JOURNAL OF PHYSIOLOGY, 1980, 239 (02) :F160-F166
[9]   SELECTIVE INHIBITORY ACTIONS OF SODIUM-PARA-BENZYL-4-[1-OXO-2-(4-CHLOROBENZYL)-3-PHENYL PROPYL] PHENYL PHOSPHONATE (N-0164) AND INDOMETHACIN ON BIOSYNTHESIS OF PROSTAGLANDINS AND THROMBOXANES FROM ARACHIDONIC-ACID [J].
EAKINS, KE ;
KULKARNI, PS .
BRITISH JOURNAL OF PHARMACOLOGY, 1977, 60 (01) :135-140
[10]   COMPARISON OF IMIDAZOLE AND 9,11-AZOPROSTA-5,13-DIENOIC ACID - 2 SELECTIVE THROMBOXANE SYNTHETASE INHIBITORS [J].
FITZPATRICK, FA ;
GORMAN, RR .
BIOCHIMICA ET BIOPHYSICA ACTA, 1978, 539 (02) :162-172