ESTERIFICATION OF N-PROTECTED ALPHA-AMINO-ACIDS WITH ALCOHOL/CARBODIIMIDE/4-(DIMETHYLAMINO)-PYRIDINE - RACEMIZATION OF ASPARTIC AND GLUTAMIC-ACID DERIVATIVES

被引：227

作者：

DHAON, MK ^{[1
]}

OLSEN, RK ^{[1
]}

RAMASAMY, K ^{[1
]}

机构：

[1] UTAH STATE UNIV,DEPT CHEM & BIOCHEM,LOGAN,UT 84322

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1982年 / 47卷 / 10期

关键词：

D O I：

10.1021/jo00349a028

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：1962 / 1965

页数：4

共 17 条

[1] TERT-BUTYL ESTERS OF AMINO ACIDS AND PEPTIDES AND THEIR USE IN PEPTIDE SYNTHESIS [J].

ANDERSON, GW ;

CALLAHAN, FM .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1960, 82 (13) :3359-3363

[2] RACEMIZATION OF ACTIVATED, URETHANE-PROTECTED AMINO-ACIDS BY PARA-DIMETHYLAMINOPYRIDINE - SIGNIFICANCE IN SOLID-PHASE PEPTIDE-SYNTHESIS [J].

ATHERTON, E ;

BENOITON, NL ;

BROWN, E ;

SHEPPARD, RC ;

WILLIAMS, BJ .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1981, (07) :336-337

[3]

Bodanszky M., 1976, PEPTIDE SYNTHESIS

[4] AMINO-ACIDS AND PEPTIDES .30. FACILITATION OF PEPTIDE SYNTHESIS BY USE OF 4-PICOLYL ESTERS FOR CARBOXY-GROUP PROTECTION [J].

CAMBLE, R ;

GARNER, R ;

YOUNG, GT .

JOURNAL OF THE CHEMICAL SOCIETY C-ORGANIC, 1969, (14) :1911-&

[5] SEPARATION OF ENANTIOMERS ON PACKED-COLUMNS CONTAINING OPTICALLY-ACTIVE DIAMIDE PHASES [J].

CHARLES, R ;

BEITLER, U ;

FEIBUSH, B ;

GILAV, E .

JOURNAL OF CHROMATOGRAPHY, 1975, 112 (OCT29) :121-133

[6]

GILON C, 1979, TETRAHEDRON LETT, P3811

[7]

HASSNER A, 1978, TETRAHEDRON LETT, P4475

[8] SEPARATION OF DIASTEREOMERS USING A LOW-COST PREPARATIVE MEDIUM-PRESSURE LIQUID CHROMATOGRAPH [J].

MEYERS, AI ;

SLADE, J ;

SMITH, RK ;

MIHELICH, ED ;

HERSHENSON, FM ;

LIANG, CD .

JOURNAL OF ORGANIC CHEMISTRY, 1979, 44 (13) :2247-2249

[9] ELIMINATION-ADDITION .16. ELIMINATION IN 2-SULPHONYLETHYL CARBOXYLATES - A METHOD FOR PROTECTION OF CARBOXY-GROUPS IN PEPTIDE SYNTHESIS [J].

MILLER, AW ;

STIRLING, CJ .

JOURNAL OF THE CHEMICAL SOCIETY C-ORGANIC, 1968, (21) :2612-&

[10]

NEISES B, 1978, ANGEW CHEM INT EDIT, V17, P552

← 1 2 →