SYNTHESIS OF 11-AZASTEROIDS FROM AROMATIC-AMINES, FORMALDEHYDE AND CYCLOPENTADIENE

被引：24

作者：

GREGOIRE, PJ ^{[1
]}

MELLOR, JM ^{[1
]}

MERRIMAN, GD ^{[1
]}

机构：

[1] UNIV SOUTHAMPTON,DEPT CHEM,SOUTHAMPTON SO9 5NH,HANTS,ENGLAND

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 48期

关键词：

D O I：

10.1016/0040-4039(91)85051-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient one pot synthesis of azasteroids and related tetrahydroquinoline skeletons has been developed by reaction of aromatic primary amines with formaldehyde and cyclopentadiene.

引用

页码：7099 / 7102

页数：4

共 8 条

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[3] ROLE REVERSAL IN THE CYCLOCONDENSATION OF CYCLOPENTADIENE WITH HETERODIENOPHILES DERIVED FROM ARYL AMINES AND ALDEHYDES - SYNTHESIS OF NOVEL TETRAHYDROQUINOLINES
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[5] HIGHLY STEREOSELECTIVE TOTAL SYNTHESES OF (+/-)-CHELIDONINE AND OF (+/-)-NORCHELIDONINE BY AN INTRAMOLECULAR ORTHO-QUINODIMETHANE NITROSTYRENE-CYCLOADDITION
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[7] PHOTOINDUCED MOLECULAR-TRANSFORMATIONS .107. A VERSATILE SUBSTITUTION OF A CARBONYL GROUP OF STEROIDAL KETONES BY A HETEROATOM - THE SYNTHESIS OF AZASTEROIDS, OXASTEROIDS, THIASTEROIDS, SELENASTEROIDS, AND TELLURASTEROIDS
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[J]. JOURNAL OF ORGANIC CHEMISTRY, 1990, 55 (07) : 2170 - 2176
[8] INTERMOLECULAR AND INTRAMOLECULAR HETERO-DIELS-ALDER REACTIONS .29. SYNTHESIS OF ENANTIOMERICALLY PURE HETEROSTEROIDS BY INTRAMOLECULAR HETERO-DIELS-ALDER REACTION
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