PHASE-I TRIAL OF TRIMETREXATE GLUCURONATE ON A 5-DAY BOLUS SCHEDULE - CLINICAL-PHARMACOLOGY AND PHARMACODYNAMICS

被引:32
作者
GROCHOW, LB
NOE, DA
DOLE, GB
ROWINSKY, EK
ETTINGER, DS
GRAHAM, ML
MCGUIRE, WP
DONEHOWER, RC
机构
关键词
D O I
10.1093/jnci/81.2.124
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:124 / 130
页数:7
相关论文
共 20 条
[1]  
BALIS FM, 1986, CANCER RES, V46, P169
[2]   2,4-DIAMINO-5-METHYL-6-[(3,4,5-TRIMETHOXYANILINO)METHYL]QUINAZOLINE (TMQ), A POTENT NON-CLASSICAL FOLATE ANTAGONIST INHIBITOR .1. EFFECT ON DIHYDROFOLATE-REDUCTASE AND GROWTH OF RODENT TUMORS INVITRO AND INVIVO [J].
BERTINO, JR ;
SAWICKI, WL ;
MOROSON, BA ;
CASHMORE, AR ;
ELSLAGER, EF .
BIOCHEMICAL PHARMACOLOGY, 1979, 28 (12) :1983-1987
[3]  
BERTINO JR, 1987, NATL CANCER I MONOGR, V5, P87
[4]  
CHABNER B, 1982, PHARM PRINCIPLES CAN, P236
[5]  
DIDDENS H, 1983, CANCER RES, V43, P5286
[6]  
DONEHOWER RC, 1985, P AN M AM SOC CLIN, V4, P32
[7]  
DRAKE JC, 1985, CANCER TREAT REP, V69, P641
[8]  
FANUCCHI MP, 1987, CANCER RES, V47, P3303
[9]   ENZYMATIC ASSAYS FOR 2,4-DIAMINO-5-METHYL-6-[(3,4,5-TRIMETHOXYANILINO)METHYL]QUINAZOLINE, A PROMISING NEW NON-CLASSICAL ANTIFOLATE [J].
HEUSNER, JJ ;
MCCORMACK, JJ .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1981, 70 (07) :827-828
[10]   CLINICAL-PHARMACOLOGY OF TRIMETREXATE [J].
HO, DHW ;
COVINGTON, WP ;
LEGHA, SS ;
NEWMAN, RA ;
KRAKOFF, IH .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1987, 42 (03) :351-356