SYNTHESIS OF 7-ALKENYLQUINOLONE, 7-CYCLOALKENYLQUINOLONE, AND 7-(1,2,3,6-TETRAHYDRO-4-PYRIDINYL)QUINOLONES

被引：16

作者：

KIELY, JS

LABORDE, E

LESHESKI, LE

BUCSH, RA

机构：

[1] Chemistry Department, Parke-Davis Pharmaceutical Research Division, Warner-Lambert Company, Ann Arbor, Michigan

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1991年 / 28卷 / 06期

关键词：

D O I：

10.1002/jhet.5570280621

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of 1-cyclopropyl-1,4-dihydro-4-oxoquinolines was prepared in which the C-7 position is substituted with a vinyl, a 1-cyclopentenyl, or a 1,2,3,6-tetrahydro-4-pyridinyl group. These quinolones were synthesized via a palladium-catalyzed cross coupling of a 7-quinolyltriflate with an appropriately functionalized vinyl-stannane.

引用

页码：1581 / 1585

页数：5

共 12 条

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