DERIVATIVES OF 3,4-DIHYDROCARBOSTYRIL AS BETA-ADRENERGIC BLOCKING-AGENTS

被引：85

作者：

NAKAGAWA, K ^{[1
]}

MURAKAMI, N ^{[1
]}

YOSHIZAK.S ^{[1
]}

TOMINAGA, M ^{[1
]}

MORI, H ^{[1
]}

YABUUCHI, Y ^{[1
]}

SHINTANI, S ^{[1
]}

机构：

[1] OTSUKA PHARM CO LTD, TOKUSHIMA FACTORY, RES LAB 1, 463-10 KAGASUNO, KAWAUCHI, TOKUSHIMA, JAPAN

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1974年 / 17卷 / 05期

关键词：

D O I：

10.1021/jm00251a013

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

The compounds were prepared and their adrenergic .beta.-receptor blocking activity was evaluated by inhibition of the depressor and the positive chronotropic responses to isoproterenol in the dog.

引用

页码：529 / 533

页数：5

共 19 条

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[6] 1-ISOPROPYLAMINO-3-(4-INDANOXY)-2-PROPANOL HCL - A POTENT BETA-ADRENOCEPTOR ANTAGONIST
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