ROLE OF ESTROGEN-RECEPTORS AND ANTIESTROGEN BINDING-SITES IN AN EARLY EFFECT OF ANTIESTROGENS, THE INHIBITION OF CHOLESTEROL-BIOSYNTHESIS

被引:22
作者
CYPRIANI, B
TABACIK, C
DESCOMPS, B
DEPAULET, AC
机构
关键词
D O I
10.1016/0022-4731(88)90284-1
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
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引用
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页码:763 / 771
页数:9
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共 44 条
[1]  
AITKEN SC, 1985, CANCER RES, V45, P1611
[2]   THE ANTIPROLIFERATIVE EFFECT OF TAMOXIFEN IN BREAST-CANCER CELLS - MEDIATION BY THE ESTROGEN-RECEPTOR [J].
BARDON, S ;
VIGNON, F ;
DEROCQ, D ;
ROCHEFORT, H .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1984, 35 (2-3) :89-96
[3]   PHENOL RED IN TISSUE-CULTURE MEDIA IS A WEAK ESTROGEN - IMPLICATIONS CONCERNING THE STUDY OF ESTROGEN-RESPONSIVE CELLS IN CULTURE [J].
BERTHOIS, Y ;
KATZENELLENBOGEN, JA ;
KATZENELLENBOGEN, BS .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (08) :2496-2500
[4]   EVIDENCE FOR BIOLOGICAL ACTION OF THE ANTI-ESTROGENS LY117018 AND TAMOXIFEN BY DIFFERENT MECHANISMS [J].
BLACK, LJ ;
GOODE, RL .
ENDOCRINOLOGY, 1981, 109 (03) :987-989
[5]   HIGH-AFFINITY BINDING TO THE ESTROGEN-RECEPTOR OF [4-HYDROXYTAMOXIFEN-H-3, AN ACTIVE ANTI-ESTROGEN METABOLITE [J].
BORGNA, JL ;
ROCHEFORT, H .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1980, 20 (01) :71-85
[6]   A DIPHENYLMETHANE DERIVATIVE SELECTIVE FOR THE ANTI-ESTROGEN BINDING-SITE MAY HELP DEFINE ITS BIOLOGICAL ROLE [J].
BRANDES, LJ .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 124 (01) :244-249
[7]  
CHEN HW, 1984, FED PROC, V43, P126
[8]   HIGH-AFFINITY CYTOSOL BINDING SITE(S) FOR ANTIESTROGENS IN 2 HUMAN-BREAST CANCER CELL-LINES AND IN BIOPSY SPECIMENS DEVOID OF ESTROGEN-RECEPTORS [J].
CHOUVET, C ;
SAEZ, S .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1984, 21 (06) :755-761
[9]   TRIPHENYLETHYLENE ANTIESTROGEN BINDING-SITES (TABS) SPECIFICITY [J].
CLARK, JH ;
MITCHELL, WC ;
GUTHRIE, SC .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1987, 26 (04) :433-437
[10]  
COEZY E, 1982, CANCER RES, V42, P317