SYNTHESIS OF 4-(2-CHLOROETHYL)-2,3-DIHYDRO[1,4]OXAZINO[2,3-B]QUINOLINE AND 4-(2-CHLOROETHYL)-2,3-DIHYDROPYRIDO[2,3-B][1,4]OXAZINE

被引：16

作者：

ANDERSON, WK

DALVIE, DK

机构：

[1] Department of Medicinal Chemistry, School of Pharmacy, State University of New York at Buffalo, Buffalo, New York

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1993年 / 30卷 / 06期

关键词：

D O I：

10.1002/jhet.5570300614

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The title compounds were synthesized from 3-[bis(2-hydroxyethyl)amino]quinolin-2(1H)-one 11a and 3-[bis(2-hydroxyethyl)amino]pyridin-2(1H)-one 18 respectively. The preparation involved a tandem chlorination/cyclization reaction.

引用

页码：1533 / 1536

页数：4

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