DESIGN, SYNTHESIS AND SOME USES OF RECEPTOR-SPECIFIC AGONISTS AND ANTAGONISTS OF VASOPRESSIN AND OXYTOCIN

被引：97

作者：

MANNING, M ^{[1
]}

SAWYER, WH ^{[1
]}

机构：

[1] COLUMBIA UNIV COLL PHYS & SURG, DEPT PHARMACOL, NEW YORK, NY 10032 USA

来源：

JOURNAL OF RECEPTOR RESEARCH | 1993年 / 13卷 / 1-4期

关键词：

D O I：

10.3109/10799899309073655

中图分类号：

Q2 [细胞生物学];

学科分类号：

071009 ; 090102 ;

摘要：

Selective agonists and antagonists are powerful tools for studies on AVP and OT receptors and on the physiological and pathophysiological roles of AVP and OT. Here we show how some of these peptides and their radiolabelled derivatives were designed. We also present examples of the currently available cyclic and linear OT and AVP agonists and antagonists from our laboratories.

引用

页码：195 / 214

页数：20

共 46 条

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