EFFECTS OF CATIONS ON BINDING, IN MEMBRANE SUSPENSIONS, OF VARIOUS OPIOIDS AT MU-SITES OF RABBIT CEREBELLUM AND KARRA-SITES OF GUINEA-PIG CEREBELLUM

被引:19
作者
KOSTERLITZ, HW
PATERSON, SJ
ROBSON, LE
TRAYNOR, JR
机构
关键词
D O I
10.1111/j.1476-5381.1987.tb10298.x
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:431 / 437
页数:7
相关论文
共 10 条
[1]   BREMAZOCINE IS AN AGONIST AT KAPPA-OPIOID RECEPTORS AND AN ANTAGONIST AT MU-OPIOID RECEPTORS IN THE GUINEA-PIG MYENTERIC PLEXUS [J].
CORBETT, AD ;
KOSTERLITZ, HW .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 89 (01) :245-249
[2]   UNEXPECTED ANTAGONISM IN THE RAT VAS-DEFERENS BY BENZOMORPHANS WHICH ARE AGONISTS IN OTHER PHARMACOLOGICAL TESTS [J].
GILLAN, MGC ;
KOSTERLITZ, HW ;
MAGNAN, J .
BRITISH JOURNAL OF PHARMACOLOGY, 1981, 72 (01) :13-15
[3]   K-BINDING AND DEGRADATION OF [H-3] DYNORPHIN-A (1-8) AND [H-3] DYNORPHIN-A (1-9) IN SUSPENSIONS OF GUINEA-PIG BRAIN MEMBRANES [J].
GILLAN, MGC ;
ROBSON, LE ;
MCKNIGHT, AT ;
KOSTERLITZ, HW .
JOURNAL OF NEUROCHEMISTRY, 1985, 45 (04) :1034-1042
[4]   SPECTRUM OF THE MU-BINDING, DELTA-BINDING AND KAPPA-BINDING SITES IN HOMOGENATES OF RAT-BRAIN [J].
GILLAN, MGC ;
KOSTERLITZ, HW .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 77 (03) :461-468
[5]  
Hill A., 1910, J PHYSIOL-LONDON, V40, piv
[6]  
MEUNIER JC, 1983, MOL PHARMACOL, V24, P23
[7]   CONTROL BY CATIONS OF OPIOID BINDING IN GUINEA-PIG BRAIN MEMBRANES [J].
PATERSON, SJ ;
ROBSON, LE ;
KOSTERLITZ, HW .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (16) :6216-6220
[8]  
PERT CB, 1974, MOL PHARMACOL, V10, P868
[9]   OPIOID BINDING-SITES OF THE KAPPA-TYPE IN GUINEA-PIG CEREBELLUM [J].
ROBSON, LE ;
FOOTE, RW ;
MAURER, R ;
KOSTERLITZ, HW .
NEUROSCIENCE, 1984, 12 (02) :621-&
[10]  
TRAYNOR JR, 1987, IN PRESS EUR J PHARM