RENIN INHIBITORS CONTAINING HYDROPHILIC GROUPS - TETRAPEPTIDES WITH ENHANCED AQUEOUS SOLUBILITY AND NANOMOLAR POTENCY

被引：47

作者：

BOCK, MG ^{[1
]}

DIPARDO, RM ^{[1
]}

EVANS, BE ^{[1
]}

FREIDINGER, RM ^{[1
]}

RITTLE, KE ^{[1
]}

PAYNE, LS ^{[1
]}

BOGER, J ^{[1
]}

WHITTER, WL ^{[1
]}

LAMONT, BI ^{[1
]}

ULM, EH ^{[1
]}

BLAINE, EH ^{[1
]}

SCHORN, TW ^{[1
]}

VEBER, DF ^{[1
]}

机构：

[1] MERCK SHARP & DOHME RES LABS, RAHWAY, NJ 07065 USA

来源：

关键词：

D O I：

10.1021/jm00118a009

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1918 / 1923

页数：6

共 34 条

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