RENIN INHIBITORS - STATINE-CONTAINING TETRAPEPTIDES WITH VARIED HYDROPHOBIC CARBOXY TERMINI

被引：15

作者：

BOCK, MG ^{[1
]}

DIPARDO, RM ^{[1
]}

EVANS, BE ^{[1
]}

RITTLE, KE ^{[1
]}

BOGER, J ^{[1
]}

POE, M ^{[1
]}

LAMONT, BI ^{[1
]}

LYNCH, RJ ^{[1
]}

ULM, EH ^{[1
]}

VLASUK, GP ^{[1
]}

GREENLEE, WJ ^{[1
]}

VEBER, DF ^{[1
]}

机构：

[1] MERCK SHARP & DOHME RES LABS, RAHWAY, NJ 07065 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 10期

关键词：

D O I：

10.1021/jm00393a029

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1853 / 1857

页数：5

共 26 条

[1] NOVEL RENIN INHIBITORS - SYNTHESIS OF AMINOSTATINE AND COMPARISON WITH STATINE-CONTAINING ANALOGS
ARROWSMITH, RJ
CARTER, K
DANN, JG
DAVIES, DE
HARRIS, CJ
MORTON, JA
LISTER, P
ROBINSON, JA
WILLIAMS, DJ
[J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1986, (10) : 755 - 757
[2] DIPEPTIDE ANALOGS - SYNTHESIS OF A POTENT RENIN INHIBITOR
BOCK, MG
DIPARDO, RM
EVANS, BE
RITTLE, KE
BOGER, JS
FREIDINGER, RM
VEBER, DF
[J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1985, (03) : 109 - 110
[3] BOGER J, 1985, REGUL PEPTIDES, P8
[4] NOVEL RENIN INHIBITORS CONTAINING THE AMINO-ACID STATINE
BOGER, J
LOHR, NS
ULM, EH
POE, M
BLAINE, EH
FANELLI, GM
LIN, TY
PAYNE, LS
SCHORN, TW
LAMONT, BI
VASSIL, TC
STABILITO, II
VEBER, DF
RICH, DH
BOPARI, AS
[J]. NATURE, 1983, 303 (5912) : 81 - 84
[5] RENIN INHIBITORS - SYNTHESES OF SUBNANOMOLAR, COMPETITIVE, TRANSITION-STATE ANALOG INHIBITORS CONTAINING A NOVEL ANALOG OF STATINE
BOGER, J
PAYNE, LS
PERLOW, DS
LOHR, NS
POE, M
BLAINE, EH
ULM, EH
SCHORN, TW
LAMONT, BI
LIN, TY
KAWAI, M
RICH, DH
VEBER, DF
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (12) : 1779 - 1790
[6] BOGER J, 1983, PEPTIDES STRUCTURE F, P569
[7] CUMIN F, 1985, J BIOL CHEM, V260, P9154
[8] THE DETERMINATION OF ENZYME INHIBITOR CONSTANTS
DIXON, M
[J]. BIOCHEMICAL JOURNAL, 1953, 55 (01) : 170 - 171
[9] ERICKSON BW, 1976, PROTEINS, V2, P257
[10] A UNIQUELY POTENT RENIN INHIBITOR AND ITS UNANTICIPATED PLASMA-BINDING COMPONENT
EVANS, BE
RITTLE, KE
BOCK, MG
BENNETT, CD
DIPARDO, RM
BOGER, J
POE, M
ULM, EH
LAMONT, BI
BLAINE, EH
FANELLI, GM
STABILITO, II
VEBER, DF
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (12) : 1755 - 1756

← 1 2 3 →